TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human MCHR1 expressed in HEK293 cells assessed as [35S]GTPgammaS accumulationMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human MCHR1 expressed in HEK293 cells assessed as [35S]GTPgammaS accumulationMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Antagonist activity at human MCHR1 expressed in HEK293 cells assessed as [35S]GTPgammaS accumulationMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human MCHR1 expressed in HEK293 cells assessed as [35S]GTPgammaS accumulationMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 142nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 144nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 173nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 313nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 339nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 417nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 444nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 597nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 815nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human ERG activation expressed in CHO cells by rubidium efflux assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair