Compile Data Set for Download or QSAR
maximum 50k data
Found 54 Enz. Inhib. hit(s) with all data for entry = 50030782
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301315(CHEMBL568467 | N-(3,4-dimethyl-5-(morpholinomethyl...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50277153(4-methyl-3-(morpholinosulfonyl)-N-((1S,2R,4R)-1,3,...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301316(CHEMBL568468 | N-(3,4-dimethyl-5-(morpholinomethyl...)
Affinity DataKi:  8.60nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301312(3,3-difluoro-2-methyl-N-(4-methyl-3-(morpholinomet...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50301306(2-methyl-N-(4-methyl-3-(morpholinomethyl)-5-(trifl...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301317(4-methyl-3-(morpholinomethyl)-N-((1S,4R)-1,3,3-tri...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301307(CHEMBL577487 | N-(2-fluoro-4-methyl-5-(morpholinom...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301318(4-methyl-3-(2-morpholinoethyl)-N-((1S,4R)-1,3,3-tr...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301319(4-methyl-3-(3-morpholinopropyl)-N-((1S,4R)-1,3,3-t...)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301313(2-methyl-N-(4-methyl-3-(morpholinomethyl)phenyl)cy...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301321(4-methyl-3-(3-morpholino-3-oxopropyl)-N-((1S,4R)-1...)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301306(2-methyl-N-(4-methyl-3-(morpholinomethyl)-5-(trifl...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301308(CHEMBL567795 | N-(2-fluoro-4-methyl-5-(morpholinom...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301314(2,2-dimethyl-N-(4-methyl-3-(morpholinomethyl)pheny...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50277153(4-methyl-3-(morpholinosulfonyl)-N-((1S,2R,4R)-1,3,...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301320(4-methyl-3-morpholino-N-((1S,4R)-1,3,3-trimethylbi...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301309(CHEMBL565515 | N-(2,4-dimethyl-5-(morpholinomethyl...)
Affinity DataKi:  440nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301315(CHEMBL568467 | N-(3,4-dimethyl-5-(morpholinomethyl...)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301310(CHEMBL567924 | N-(2,4-dimethyl-5-(morpholinomethyl...)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301316(CHEMBL568468 | N-(3,4-dimethyl-5-(morpholinomethyl...)
Affinity DataKi:  540nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301322(4-methyl-3-(2-morpholino-2-oxoethyl)-N-(1,3,3-trim...)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301317(4-methyl-3-(morpholinomethyl)-N-((1S,4R)-1,3,3-tri...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301323(4-methyl-3-(morpholine-4-carbonyl)-N-((1S,4R)-1,3,...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301318(4-methyl-3-(2-morpholinoethyl)-N-((1S,4R)-1,3,3-tr...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301313(2-methyl-N-(4-methyl-3-(morpholinomethyl)phenyl)cy...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301321(4-methyl-3-(3-morpholino-3-oxopropyl)-N-((1S,4R)-1...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301319(4-methyl-3-(3-morpholinopropyl)-N-((1S,4R)-1,3,3-t...)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301322(4-methyl-3-(2-morpholino-2-oxoethyl)-N-(1,3,3-trim...)
Affinity DataKi:  3.90E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301323(4-methyl-3-(morpholine-4-carbonyl)-N-((1S,4R)-1,3,...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301312(3,3-difluoro-2-methyl-N-(4-methyl-3-(morpholinomet...)
Affinity DataKi:  6.30E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301320(4-methyl-3-morpholino-N-((1S,4R)-1,3,3-trimethylbi...)
Affinity DataKi:  9.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301319(4-methyl-3-(3-morpholinopropyl)-N-((1S,4R)-1,3,3-t...)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301318(4-methyl-3-(2-morpholinoethyl)-N-((1S,4R)-1,3,3-tr...)
Affinity DataEC50:  64nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301317(4-methyl-3-(morpholinomethyl)-N-((1S,4R)-1,3,3-tri...)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50277153(4-methyl-3-(morpholinosulfonyl)-N-((1S,2R,4R)-1,3,...)
Affinity DataEC50:  6.60nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301316(CHEMBL568468 | N-(3,4-dimethyl-5-(morpholinomethyl...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301315(CHEMBL568467 | N-(3,4-dimethyl-5-(morpholinomethyl...)
Affinity DataEC50:  5.5nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301314(2,2-dimethyl-N-(4-methyl-3-(morpholinomethyl)pheny...)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301313(2-methyl-N-(4-methyl-3-(morpholinomethyl)phenyl)cy...)
Affinity DataEC50:  76nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301312(3,3-difluoro-2-methyl-N-(4-methyl-3-(morpholinomet...)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301310(CHEMBL567924 | N-(2,4-dimethyl-5-(morpholinomethyl...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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