Compile Data Set for Download or QSAR
maximum 50k data
Found 29 Enz. Inhib. hit(s) with all data for entry = 50030928
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50270528(3-BROMO-7-NITROINDAZOLE | 3-bromo-7-nitro-1H-indaz...)
Affinity DataIC50:  170nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50270528(3-BROMO-7-NITROINDAZOLE | 3-bromo-7-nitro-1H-indaz...)
Affinity DataIC50:  290nMAssay Description:Inhibition of NOS2More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50304142(2,7-dinitro-2H-indazole | CHEMBL593105)
Affinity DataIC50:  620nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50209245(CHEMBL247378)
Affinity DataIC50:  710nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50209241(4-bromo-1H-indazole | CHEMBL246393)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50304143(4-nitro-1H-indazole | CHEMBL393456)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50304142(2,7-dinitro-2H-indazole | CHEMBL593105)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of NOS2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50209244(7-chloro-1H-indazole | CHEMBL247367)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50209237(6-bromo-1H-indazole | CHEMBL247365)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50209245(CHEMBL247378)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of NOS2More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50209239(7-bromo-1H-indazole | CHEMBL439566)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50209235(4-iodo-1H-indazole | CHEMBL246534)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50209236(6-Chloro-1H-indazole | CHEMBL392184)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50284964(6-NITROINDAZOLE | 6-Nitro-1H-indazole | CHEMBL5427...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50209243(5-iodo-1H-indazole | CHEMBL391348)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50209234(4-chloro-1H-indazole | CHEMBL246533)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50304144(5-NITROINDAZOLE | 5-Nitro-1H-indazole | CHEMBL1653...)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50209242(5-chloro-1H-indazole | CHEMBL246746)
Affinity DataIC50:  5.90E+4nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50099398(5-Bromo-1H-indazole | CHEMBL16425 | cid_761929)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50304147(3-chloro-1H-indazole | CHEMBL596385)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant NOS1 assessed as citrulline formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50271275(1H-Indazol-7-amine | 1H-indazol-7-amine, 1 | CHEMB...)
Affinity DataIC50:  1.15E+5nMAssay Description:Inhibition of recombinant NOS1 assessed as citrulline formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50304145(3-chloro-6-nitro-1H-indazole | CHEMBL596229)
Affinity DataIC50:  1.58E+5nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM24627(1H-indazole | Indazole, 5 | Indazole, 6)
Affinity DataIC50:  1.78E+5nMAssay Description:Inhibition of recombinant NOS1 assessed as citrulline formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50304150(3-bromo-1,5-dinitro-1H-indazole | CHEMBL596341)
Affinity DataIC50:  2.75E+5nMAssay Description:Inhibition of recombinant NOS1 assessed as citrulline formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50304146(3-ethyl-1H-indazole | CHEMBL595903)
Affinity DataIC50:  3.10E+5nMAssay Description:Inhibition of recombinant NOS1 assessed as citrulline formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50304151(4,5,6,7-tetrafluoro-3-perfluorophenyl-1H-indazole ...)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibition of NOS2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50304148(1H-Indazol-5-ylamine | 1H-indazol-5-amine | CHEMBL...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant NOS1 assessed as citrulline formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50008990(1,2-Dihydro-indazol-3-one | 1H-indazol-3-ol | CHEM...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant NOS1 assessed as citrulline formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Uned

Curated by ChEMBL
LigandPNGBDBM50304149(1H-indazol-6-amine | CHEMBL594707 | cid_81423)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant NOS1 assessed as citrulline formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed