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Found 8 Enz. Inhib. hit(s) with all data for entry = 50030945
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM22594(7-methoxy-4-nitro-5-oxatricyclo[7.4.0.0^{2,6}]trid...)
Affinity DataEC50:  1.47E+3nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304336(2-Nitro-naphtho[2,1-b]furan-7-ol | 2-nitronaphtho[...)
Affinity DataEC50:  1.95E+3nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304337(2-(2-Nitro-naphtho[2,1-b]furan-1-yl)-ethanol | 2-(...)
Affinity DataEC50:  1.22E+3nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304342(CHEMBL611816 | naphtho[2,1-b]furan-2-carboxamide)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304339(8-Methoxy-2-nitro-naphtho[2,1-b]furan | 8-methoxy-...)
Affinity DataEC50:  2.33E+3nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304340(2-Nitro-naphtho[2,1-b]furan | 2-nitronaphtho[2,1-b...)
Affinity DataEC50:  2.09E+3nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304341(7-Methoxy-2-nitro-naphtho[2,1-b]furan | 7-methoxy-...)
Affinity DataEC50:  2.57E+3nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304338(1-Methyl-2-nitro-naphtho[2,1-b]furan | 1-methyl-2-...)
Affinity DataEC50:  1.28E+3nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed