Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50030741
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300767(CHEMBL570566 | {[(9Z)-octadec-9-en-1-yl]sulfamoyl}...)
Affinity DataKi:  1.89E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300765(CHEMBL583108 | N-(cis-5-cis-8-cis-11-cis-14-eicosa...)
Affinity DataKi:  2.34E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300770(CHEMBL568489 | N-(cis-5-cis-8-cis-11-cis-14-eicosa...)
Affinity DataKi:  4.01E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300769(CHEMBL374746 | N-(1-adamantyl)-N'-propylsulfamide)
Affinity DataKi:  4.23E+3nMAssay Description:Displacement of [3H]WIN55212-2 from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300771(CHEMBL570988 | N-(cis-9-cis-12-octadecadienyl)sulf...)
Affinity DataKi:  6.41E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50202584(CHEMBL218643 | N-(2-adamantyl)-N'-propylsulfamide)
Affinity DataKi:  6.67E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300766(CHEMBL569658 | N-(cis-9-cis-12-octadecadienyl)-N'-...)
Affinity DataKi:  7.19E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300769(CHEMBL374746 | N-(1-adamantyl)-N'-propylsulfamide)
Affinity DataKi:  8.58E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50202583(CHEMBL219156 | N-octadecyl-N'-propylsulfamide)
Affinity DataKi:  9.10E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50202583(CHEMBL219156 | N-octadecyl-N'-propylsulfamide)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]WIN55212-2 from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50202584(CHEMBL218643 | N-(2-adamantyl)-N'-propylsulfamide)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]WIN55212-2 from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50202579(CHEMBL218794 | N-octadecylsulfamide)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300764(CHEMBL571044 | N-oleyl-N'-propylsulfamide)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300768(CHEMBL437157 | N-(1-(1-adamantyl)ethyl)-N'-propyls...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300768(CHEMBL437157 | N-(1-(1-adamantyl)ethyl)-N'-propyls...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]WIN55212-2 from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed