Affinity DataKi: 7nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.80nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibition of JAK2-mediated STAT5 phosphorylation in GMCSF-stimulated human TF1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 86nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of JAK2-mediated STAT5 phosphorylation in GMCSF-stimulated human TF1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair