Compile Data Set for Download or QSAR
maximum 50k data
Found 66 Enz. Inhib. hit(s) with all data for entry = 50041787
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415550(CHEMBL599760 | Ro-85)
Affinity DataIC50:  31.6nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415553(CHEMBL605130)
Affinity DataIC50:  39.8nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415601(CHEMBL598103)
Affinity DataIC50:  39.8nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415574(CHEMBL597486)
Affinity DataIC50:  50.1nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415599(CHEMBL604740)
Affinity DataIC50:  63.1nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415564(CHEMBL598728)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415550(CHEMBL599760 | Ro-85)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415575(CHEMBL597485)
Affinity DataIC50:  126nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415583(CHEMBL597110)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415563(CHEMBL605325)
Affinity DataIC50:  251nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415566(CHEMBL604571)
Affinity DataIC50:  398nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415578(CHEMBL603453)
Affinity DataIC50:  398nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415550(CHEMBL599760 | Ro-85)
Affinity DataIC50:  398nMAssay Description:Antagonist activity at human P2X3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415593(CHEMBL599348)
Affinity DataIC50:  501nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415577(CHEMBL597480)
Affinity DataIC50:  501nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415576(CHEMBL597285)
Affinity DataIC50:  501nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415571(CHEMBL598498)
Affinity DataIC50:  501nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415586(CHEMBL603254)
Affinity DataIC50:  631nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415569(CHEMBL605156)
Affinity DataIC50:  631nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415596(CHEMBL596814)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415597(CHEMBL598729)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415587(CHEMBL598865)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415588(CHEMBL605322)
Affinity DataIC50:  1.26E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415581(CHEMBL597316)
Affinity DataIC50:  1.26E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415580(CHEMBL598471)
Affinity DataIC50:  1.26E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415570(CHEMBL590972)
Affinity DataIC50:  1.26E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415572(CHEMBL598497)
Affinity DataIC50:  1.58E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415584(CHEMBL591530)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415592(CHEMBL599335)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415573(CHEMBL604725)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415595(CHEMBL602338)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415555(CHEMBL597016)
Affinity DataIC50:  2.51E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415565(CHEMBL605346)
Affinity DataIC50:  2.51E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415585(CHEMBL601912)
Affinity DataIC50:  3.98E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415579(CHEMBL597061)
Affinity DataIC50:  5.01E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415582(CHEMBL597111)
Affinity DataIC50:  5.01E+3nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415557(CHEMBL599738)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415558(CHEMBL599739)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415559(CHEMBL599757)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415560(CHEMBL605126)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415561(CHEMBL597899)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415562(CHEMBL604944)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415563(CHEMBL605325)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415563(CHEMBL605325)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415563(CHEMBL605325)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 5(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415563(CHEMBL605325)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 6(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415563(CHEMBL605325)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415563(CHEMBL605325)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415567(CHEMBL600997)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50415568(CHEMBL600996)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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