TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Binding affinity to pregnane receptor in human hepatocytesMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Affinity DataKi: 372nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Affinity DataKi: 4.06E+3nMAssay Description:Binding affinity to adrenergic alpha2c receptorMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Affinity DataKi: 7.85E+3nMAssay Description:Binding affinity to dopamine D4 receptorMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Affinity DataKi: 9.34E+3nMAssay Description:Binding affinity to adrenergic alpha2A receptorMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Affinity DataKi: 9.64E+3nMAssay Description:Binding affinity to adrenergic alpha2c receptorMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of CRF1 receptorMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Westfalische Wilhelms-Universitat
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant CRF1 receptor expressed in CHO cells assessed as inhibition of CRF-induced cAMP formationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair