Compile Data Set for Download or QSAR
maximum 50k data
Found 94 Enz. Inhib. hit(s) with all data for entry = 50032423
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  1.18nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328956(CHEMBL1269774 | N-{11-[(11-Aminoundecyl)amino]unde...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328952(CHEMBL1269766 | N,N'-(Iminodiheptane-7,1-diyl)bis[...)
Affinity DataKi:  4.41nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328956(CHEMBL1269774 | N-{11-[(11-Aminoundecyl)amino]unde...)
Affinity DataKi:  4.56nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328957(CHEMBL1269773 | N-{9-[(9-Aminononyl)amino]nonyl}-5...)
Affinity DataKi:  5.44nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328967(CHEMBL1269776 | N-{11-[(11-Aminoundecyl)(methyl)am...)
Affinity DataKi:  5.51nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328960(CHEMBL1269775 | N-{9-[(9-Aminononyl)(methyl)amino]...)
Affinity DataKi:  6.12nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  6.18nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328966(CHEMBL1269769 | N,N'-[(Methylimino)dipentane-5,1-d...)
Affinity DataKi:  6.35nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328960(CHEMBL1269775 | N-{9-[(9-Aminononyl)(methyl)amino]...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328952(CHEMBL1269766 | N,N'-(Iminodiheptane-7,1-diyl)bis[...)
Affinity DataKi:  12.3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328957(CHEMBL1269773 | N-{9-[(9-Aminononyl)amino]nonyl}-5...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328967(CHEMBL1269776 | N-{11-[(11-Aminoundecyl)(methyl)am...)
Affinity DataKi:  14.7nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328961(CHEMBL1270662 | N-{7-[(7-Aminoheptyl)(methyl)amino...)
Affinity DataKi:  15.5nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328965(CHEMBL1269770 | N,N'-[(Methylimino)diheptane-7,1-d...)
Affinity DataKi:  17.3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328958(CHEMBL1270463 | N-{7-[(7-Aminoheptyl)amino]heptyl}...)
Affinity DataKi:  19.5nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328965(CHEMBL1269770 | N,N'-[(Methylimino)diheptane-7,1-d...)
Affinity DataKi:  27.5nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328953(CHEMBL1269765 | N,N'-(Iminodipentane-5,1-diyl)bis[...)
Affinity DataKi:  30.4nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328950(CHEMBL1269768 | N,N'-(Iminodiundecane-11,1-diyl)bi...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328961(CHEMBL1270662 | N-{7-[(7-Aminoheptyl)(methyl)amino...)
Affinity DataKi:  37.5nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328966(CHEMBL1269769 | N,N'-[(Methylimino)dipentane-5,1-d...)
Affinity DataKi:  38.7nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328954(CHEMBL1269019 | N,N'-(Iminodipropane-3,1-diyl)bis[...)
Affinity DataKi:  41.9nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328958(CHEMBL1270463 | N-{7-[(7-Aminoheptyl)amino]heptyl}...)
Affinity DataKi:  46.7nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328951(CHEMBL1269767 | N,N'-(Iminodinonane-9,1-diyl)bis[5...)
Affinity DataKi:  54.1nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328951(CHEMBL1269767 | N,N'-(Iminodinonane-9,1-diyl)bis[5...)
Affinity DataKi:  57.4nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328953(CHEMBL1269765 | N,N'-(Iminodipentane-5,1-diyl)bis[...)
Affinity DataKi:  68.1nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328962(CHEMBL1270563 | N-{5-[(5-Aminopentyl)(methyl)amino...)
Affinity DataKi:  88.8nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328955(CHEMBL1269764 | N,N'-(Iminodiethane-2,1-diyl)bis[5...)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328964(CHEMBL1269771 | N,N'-[(Methylimino)dinonane-9,1-di...)
Affinity DataKi:  94.1nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328950(CHEMBL1269768 | N,N'-(Iminodiundecane-11,1-diyl)bi...)
Affinity DataKi:  99.3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328962(CHEMBL1270563 | N-{5-[(5-Aminopentyl)(methyl)amino...)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328954(CHEMBL1269019 | N,N'-(Iminodipropane-3,1-diyl)bis[...)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328955(CHEMBL1269764 | N,N'-(Iminodiethane-2,1-diyl)bis[5...)
Affinity DataKi:  229nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328959(CHEMBL1270369 | N-{5-[(5-Aminopentyl)amino]pentyl}...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328964(CHEMBL1269771 | N,N'-[(Methylimino)dinonane-9,1-di...)
Affinity DataKi:  247nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328960(CHEMBL1269775 | N-{9-[(9-Aminononyl)(methyl)amino]...)
Affinity DataKi:  265nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328956(CHEMBL1269774 | N-{11-[(11-Aminoundecyl)amino]unde...)
Affinity DataKi:  305nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  313nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328959(CHEMBL1270369 | N-{5-[(5-Aminopentyl)amino]pentyl}...)
Affinity DataKi:  349nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328957(CHEMBL1269773 | N-{9-[(9-Aminononyl)amino]nonyl}-5...)
Affinity DataKi:  419nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328967(CHEMBL1269776 | N-{11-[(11-Aminoundecyl)(methyl)am...)
Affinity DataKi:  426nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328953(CHEMBL1269765 | N,N'-(Iminodipentane-5,1-diyl)bis[...)
Affinity DataKi:  451nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328954(CHEMBL1269019 | N,N'-(Iminodipropane-3,1-diyl)bis[...)
Affinity DataKi:  496nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328969(CHEMBL1270270 | N-{2-[(2-Aminoethyl)amino]ethyl}-5...)
Affinity DataKi:  506nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328952(CHEMBL1269766 | N,N'-(Iminodiheptane-7,1-diyl)bis[...)
Affinity DataKi:  553nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328958(CHEMBL1270463 | N-{7-[(7-Aminoheptyl)amino]heptyl}...)
Affinity DataKi:  622nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328965(CHEMBL1269770 | N,N'-[(Methylimino)diheptane-7,1-d...)
Affinity DataKi:  683nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328966(CHEMBL1269769 | N,N'-[(Methylimino)dipentane-5,1-d...)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328969(CHEMBL1270270 | N-{2-[(2-Aminoethyl)amino]ethyl}-5...)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328955(CHEMBL1269764 | N,N'-(Iminodiethane-2,1-diyl)bis[5...)
Affinity DataKi:  1.29E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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