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Found 26 Enz. Inhib. hit(s) with all data for entry = 50032555
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330962(2-(3,4-Dihydroxyphenyl)-7-hydroxy-4-oxo-4H-chromen...)
Affinity DataEC50:  5.37E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330986(2-(3-ethoxy-4-hydroxyphenyl)-5,7-dihydro-xy-4H-chr...)
Affinity DataEC50:  1.29E+4nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330964(2-(3,4-dihydroxyphenyl)-7-hydroxy-4-oxo-4H-chromen...)
Affinity DataEC50:  1.82E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330965(2-(3,4-dihydroxyphenyl)-7-hydroxy-4-oxo-4H-chromen...)
Affinity DataEC50:  46nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330966(2-(3,4-dihydroxyphenyl)-7-hydroxy-4-oxo-4H-chromen...)
Affinity DataEC50:  869nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330967(2-(3,4-dihydroxyphenyl)-7-hydroxy-4-oxo-4H-chromen...)
Affinity DataEC50:  2.71E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330968(2-(3,4-dihydroxyphenyl)-7-hydroxy-4-oxo-4H-chromen...)
Affinity DataEC50:  8.56E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330969(2-(3,4-dihydroxyphenyl)-7-hydroxy-4-oxo-4H-chromen...)
Affinity DataEC50:  1.12E+4nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330970(2-(3,4-dihydroxyphenyl)-7-hydroxy-4-oxo-4H-chromen...)
Affinity DataEC50:  6.92E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330971(2-(3,4-dihydroxyphenyl)-7-hydroxy-5-meth-oxy-4H-ch...)
Affinity DataEC50:  4.35E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330972(2-(3,4-Dihydroxyphenyl)-5-ethoxy-7-hydroxyl-4H-chr...)
Affinity DataEC50:  2.21E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330973(2-(3,4-dihydroxyphenyl)-7-hydroxy-5-pro-poxy-4H-ch...)
Affinity DataEC50:  3.07E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330974(2-(3,4-dihydroxyphenyl)-7-hydroxy-5-iso-propoxy-4H...)
Affinity DataEC50:  5.43E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330975(5-butoxy-2-(3,4-dihydroxyphenyl)-7-hydro-xy-4H-chr...)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330976(2-(3,4-dihydroxyphenyl)-7-hydroxy-5-isobu-toxy-4H-...)
Affinity DataEC50:  4.80E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330977(2-(3,4-dihydroxyphenyl)-7-hydroxy-5-(iso-pentyloxy...)
Affinity DataEC50:  3.43E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330978(2-(3,4-dihydroxyphenyl)-5-(hexyloxy)-7-hy-droxy-4H...)
Affinity DataEC50:  4.58E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330979(2-(3,4-dihydroxyphenyl)-7-hydroxy-5-(octy-loxy)-4H...)
Affinity DataEC50:  1.65E+4nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330980(5-(decyloxy)-2-(3,4-dihydroxyphenyl)-7-hy-droxy-4H...)
Affinity DataEC50:  3.30E+4nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330981(2-(3,4-dihydroxyphenyl)-7-hydroxy-5-(4-ph-enylbuto...)
Affinity DataEC50:  2.59E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataEC50:  1.45E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330982(2-(3,4-Dihydroxyphenyl)-5-hydroxy-4-oxo-4H-chromen...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330983(2-(3,4-dihydroxyphenyl)-5-hydroxy-4-oxo-4H-chromen...)
Affinity DataEC50:  1.69E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330984(2-(3,4-dihydroxyphenyl)-5-hydroxy-4-oxo-4H-chromen...)
Affinity DataEC50:  1.38E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330985(2-(3,4-Dihydroxyphenyl)-5,7-dimethoxy-4H-chromen-4...)
Affinity DataEC50:  3.42E+3nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50330963(2-(3,4-dihydroxyphenyl)-7-hydroxy-4-oxo-4H-chromen...)
Affinity DataEC50:  3.10E+4nMAssay Description:Agonist activity at rat DAT expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed