Compile Data Set for Download or QSAR
maximum 50k data
Found 39 Enz. Inhib. hit(s) with all data for entry = 50033353
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343731((R)-N-alpha-(2,2-Diphenylacetyl)-N-(4-ureidomethyl...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50060728((R)-2-(2,2-diphenylacetamido)-5-guanidino-N-(4-hyd...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343733((R)-N-omega-[(4-Aminobutyl)aminocarbonyl]-Na-(2,2-...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50060728((R)-2-(2,2-diphenylacetamido)-5-guanidino-N-(4-hyd...)
Affinity DataKi:  5.10nMAssay Description:Displacement of radiolabled NPY from human Y1R expressed in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343738(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343732((R)-N-omega-(6-Aminohexanoyl)-Na-(2,2-diphenylacet...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343729(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343729(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343735(1-(6-(Amino((R)-4-(2,2-diphenylacetamido)-5-oxo-5-...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343741(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343730(1-(6-((Z)-amino((R)-4-(2,2-diphenylacetamido)-5-(4...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343734((R)-5-(3-(4-aminobutyl)-1-carbamimidoylureido)-2-(...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343736(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343746(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343740(1-(6-(Amino((R)-4-(2,2-diphenylacetamido)-5-(4-hyd...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343749(1-((R)-9-Amino-24-((R)-9-amino-4-(2,2-diphenylacet...)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343747(1-((R)-9-Amino-20-((R)-9-amino-4-(2,2-diphenylacet...)
Affinity DataKi:  61nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343743(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343737(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343748(1-((R)-9-Amino-22-((R)-9-amino-4-(2,2-diphenylacet...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343744(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343745(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343739(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343742(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi: >400nMAssay Description:Displacement of Dy-635-pNPY from human Y5R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi: >500nMAssay Description:Displacement of Dy-635-pNPY from human Y2R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi: >500nMAssay Description:Displacement of Cy5-[K4]-hpp from human Y4R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343729(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of Cy5-[K4]-hpp from human Y4R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343729(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of Dy-635-pNPY from human Y2R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343729(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of Dy-635-pNPY from human Y5R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of Dy-635-pNPY from human Y5R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of Cy5-[K4]-hpp from human Y4R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of Dy-635-pNPY from human Y2R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343729(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of Cy5-[K4]-hpp from human Y4R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343729(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of Dy-635-pNPY from human Y2R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343729(1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of Dy-635-pNPY from human Y5R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKd:  5nMAssay Description:Binding affinity at Y1R in human MCF-7 cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed