Compile Data Set for Download or QSAR
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Found 6 Enz. Inhib. hit(s) with all data for entry = 50033437
TargetEstrogen receptor(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataIC50:  18nMAssay Description:Inhibition of fluorescence-labeled 17beta-estradiol binding to ERalpha receptor after 2 hrs by fluorometric analysisMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50345338((E)-1-(2,4-dihydroxy-3-((Z)-3-hydroxy-3-methylbut-...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of fluorescence-labeled 17beta-estradiol binding to ERalpha receptor after 2 hrs by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50345337(2,3-Dihydro-7-hydroxy-8-[(Z)-3-hydroxy-3-methylbut...)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of fluorescence-labeled 17beta-estradiol binding to ERalpha receptor after 2 hrs by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50345339(1-beta-Hydroxy-6,7R-dihydroxyeudesm-4(15)-ene | CH...)
Affinity DataIC50:  2.80E+6nMAssay Description:Inhibition of fluorescence-labeled 17beta-estradiol binding to ERalpha receptor after 2 hrs by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50345336((S,Z)-7-hydroxy-8-(3-hydroxy-3-methylbut-1-enyl)-5...)
Affinity DataIC50:  3.50E+6nMAssay Description:Inhibition of fluorescence-labeled 17beta-estradiol binding to ERalpha receptor after 2 hrs by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50345340((+)-Pisatin | CHEMBL1784262)
Affinity DataIC50: >5.00E+6nMAssay Description:Inhibition of fluorescence-labeled 17beta-estradiol binding to ERalpha receptor after 2 hrs by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed