Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50033441
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345471((R)-N-((S)-1-((6S,9S,12R,13R,Z)-3-ethylidene-9-iso...)
Affinity DataIC50:  2.27E+5nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345471((R)-N-((S)-1-((6S,9S,12R,13R,Z)-3-ethylidene-9-iso...)
Affinity DataIC50:  2.27E+5nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345472(CHEMBL1784750 | Nobilamide B)
Affinity DataIC50:  2.75E+5nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345472(CHEMBL1784750 | Nobilamide B)
Affinity DataIC50:  2.75E+5nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345473((R)-2-((R)-2-acetamido-3-phenylpropanamido)-N-((S)...)
Affinity DataIC50:  1.32E+6nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345473((R)-2-((R)-2-acetamido-3-phenylpropanamido)-N-((S)...)
Affinity DataIC50:  1.32E+6nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345474(CHEMBL1784749 | Nobilamide A)
Affinity DataIC50:  1.67E+6nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345474(CHEMBL1784749 | Nobilamide A)
Affinity DataIC50:  1.67E+6nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed