Affinity DataIC50: 11.5nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 13.8nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 14.4nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 14.8nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 14.8nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 15.8nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 16.6nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 16.6nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 17.8nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 18.2nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 18.2nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 18.6nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium productio...More data for this Ligand-Target Pair
Affinity DataIC50: 19.9nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 19.9nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 20.9nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 20.9nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 21.4nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium productio...More data for this Ligand-Target Pair
Affinity DataIC50: 21.9nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 24.0nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 24.0nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 26.9nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 27.5nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 28.2nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 28.2nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 29.5nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 30.2nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 31.6nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 31.6nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 38.9nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 39.8nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 40.7nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 42.7nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium productio...More data for this Ligand-Target Pair
Affinity DataIC50: 43.6nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium productio...More data for this Ligand-Target Pair
Affinity DataIC50: 45.7nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium productio...More data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium productio...More data for this Ligand-Target Pair
Affinity DataIC50: 55.0nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium productio...More data for this Ligand-Target Pair
Affinity DataIC50: 55.0nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 55.0nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 56.2nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium productio...More data for this Ligand-Target Pair
Affinity DataIC50: 56.2nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium productio...More data for this Ligand-Target Pair
Affinity DataIC50: 58.9nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium productio...More data for this Ligand-Target Pair
Affinity DataIC50: 69.2nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium productio...More data for this Ligand-Target Pair
Affinity DataIC50: 69.2nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium productio...More data for this Ligand-Target Pair
Affinity DataIC50: 70.8nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 72.4nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium productio...More data for this Ligand-Target Pair
Affinity DataIC50: 74.1nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 74.1nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 75.9nMAssay Description:Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium productio...More data for this Ligand-Target Pair
Affinity DataIC50: 77.6nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair
Affinity DataIC50: 87.1nMAssay Description:Antagonist activity at human recombinant P2X7 receptor expressed in HEK293 cells assessed as inhibition of benzoylbenzoic ATP-induced calcium product...More data for this Ligand-Target Pair