Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 50033759
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350777(CHEMBL1818827)
Affinity DataIC50:  100nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350788(CHEMBL1818826)
Affinity DataIC50:  320nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350785(CHEMBL1818829)
Affinity DataIC50:  390nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350786(CHEMBL1818828)
Affinity DataIC50:  390nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350776(CHEMBL1818825)
Affinity DataIC50:  720nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350775(CHEMBL1818824)
Affinity DataIC50:  1.25E+3nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350782(CHEMBL1818835)
Affinity DataIC50:  2.15E+3nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350774(CHEMBL1818823)
Affinity DataIC50:  2.19E+3nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350772(CHEMBL1818821)
Affinity DataIC50:  2.49E+3nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350773(CHEMBL1818822)
Affinity DataIC50:  2.70E+3nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350787(CHEMBL1818830)
Affinity DataIC50:  5.43E+3nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350780(CHEMBL1818833)
Affinity DataIC50:  8.10E+3nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350783(CHEMBL1818836)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350784(CHEMBL1818837)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350779(CHEMBL1818832)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350778(CHEMBL1818831)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350781(CHEMBL1818834)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to human ERG by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed