Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50033901
TargetBromodomain-containing protein 2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353596(CHEMBL1828986)
Affinity DataIC50:  1.60E+3nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD2 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353595(CHEMBL1828985)
Affinity DataIC50:  2.30E+3nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD2 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353588(CHEMBL1828978)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of first bromodomain of BRD2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353593(CHEMBL1828983)
Affinity DataIC50:  3.30E+3nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD2 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353588(CHEMBL1828978)
Affinity DataIC50:  3.40E+3nMAssay Description:Displacement of H3K56Ac from human CREBBP by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353592(CHEMBL1828982)
Affinity DataIC50:  4.20E+3nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD2 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353596(CHEMBL1828986)
Affinity DataIC50:  4.80E+3nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD4 by peptide displacement assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353588(CHEMBL1828978)
Affinity DataIC50:  4.80E+3nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD4 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353590(CHEMBL1828980)
Affinity DataIC50:  6.00E+3nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD2 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353588(CHEMBL1828978)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of first bromodomain of BRD4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353591(CHEMBL1828981)
Affinity DataIC50:  7.40E+3nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD2 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353595(CHEMBL1828985)
Affinity DataIC50:  7.50E+3nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD4 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353593(CHEMBL1828983)
Affinity DataIC50:  7.70E+3nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD4 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353592(CHEMBL1828982)
Affinity DataIC50:  9.70E+3nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD4 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353595(CHEMBL1828985)
Affinity DataIC50:  1.29E+4nMAssay Description:Displacement of H3K56Ac from human CREBBP by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353591(CHEMBL1828981)
Affinity DataIC50:  2.32E+4nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD4 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353590(CHEMBL1828980)
Affinity DataIC50:  2.46E+4nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD4 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353596(CHEMBL1828986)
Affinity DataIC50:  2.81E+4nMAssay Description:Displacement of H3K56Ac from human CREBBP by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353594(CHEMBL1828984)
Affinity DataIC50:  2.82E+4nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD2 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353594(CHEMBL1828984)
Affinity DataIC50:  3.22E+4nMAssay Description:Displacement of H3K56Ac from human CREBBP by peptide displacement assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353589(CHEMBL1828979)
Affinity DataIC50:  3.43E+4nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD2 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353592(CHEMBL1828982)
Affinity DataIC50:  4.54E+4nMAssay Description:Displacement of H3K56Ac from human CREBBP by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353593(CHEMBL1828983)
Affinity DataIC50:  4.94E+4nMAssay Description:Displacement of H3K56Ac from human CREBBP by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353594(CHEMBL1828984)
Affinity DataIC50:  5.12E+4nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD4 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353590(CHEMBL1828980)
Affinity DataIC50:  5.57E+4nMAssay Description:Displacement of H3K56Ac from human CREBBP by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353589(CHEMBL1828979)
Affinity DataIC50:  8.42E+4nMAssay Description:Displacement of H4Ac4 peptide from first bromodomain of human BRD4 by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353591(CHEMBL1828981)
Affinity DataIC50:  8.69E+4nMAssay Description:Displacement of H3K56Ac from human CREBBP by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353589(CHEMBL1828979)
Affinity DataIC50: >2.00E+5nMAssay Description:Displacement of H3K56Ac from human CREBBP by peptide displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353587(CHEMBL12543)
Affinity DataIC50:  2.30E+6nMAssay Description:Inhibition of CREBBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50353587(CHEMBL12543)
Affinity DataIC50:  3.40E+7nMAssay Description:Inhibition of BAZ2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed