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Found 28 Enz. Inhib. hit(s) with all data for entry = 50039738
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383074(CHEMBL2031520)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383073(CHEMBL2031521)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383076(CHEMBL2031518)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383077(CHEMBL2031516)
Affinity DataEC50:  7.10E+3nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383078(CHEMBL2031515)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383079(CHEMBL2031314)
Affinity DataEC50:  670nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383080(CHEMBL2031531)
Affinity DataEC50:  1.10E+4nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human ERbeta expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383066(CHEMBL2031529)
Affinity DataEC50:  800nMAssay Description:Agonist activity at human ERbeta expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383067(CHEMBL2031528)
Affinity DataEC50:  1.40E+4nMAssay Description:Agonist activity at human ERbeta expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383073(CHEMBL2031521)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human ERbeta expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383076(CHEMBL2031518)
Affinity DataEC50:  4.40E+3nMAssay Description:Agonist activity at human ERbeta expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383069(CHEMBL2031525)
Affinity DataEC50:  760nMAssay Description:Agonist activity at human ERbeta expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383060(CHEMBL2031539)
Affinity DataEC50:  5.50E+3nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383061(CHEMBL2029370)
Affinity DataEC50:  770nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383062(CHEMBL2031534)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383063(CHEMBL2031533)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383064(CHEMBL2031532)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383065(CHEMBL2031530)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383066(CHEMBL2031529)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383067(CHEMBL2031528)
Affinity DataEC50:  9.20nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383068(CHEMBL2031527)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383069(CHEMBL2031525)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383070(CHEMBL2031524)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383071(CHEMBL2031523)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383072(CHEMBL2031522)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50383075(CHEMBL2031519)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human ERalpha expressed in HepG2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed