Compile Data Set for Download or QSAR
maximum 50k data
Found 55 Enz. Inhib. hit(s) with all data for entry = 50040140
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389761(CHEMBL2070098)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389760(CHEMBL2070097)
Affinity DataIC50:  190nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389753(CHEMBL2070095)
Affinity DataIC50:  300nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389760(CHEMBL2070097)
Affinity DataIC50:  310nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389767(CHEMBL2070236)
Affinity DataIC50:  430nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389752(CHEMBL2070096)
Affinity DataIC50:  460nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389761(CHEMBL2070098)
Affinity DataIC50:  660nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389751(CHEMBL2070238)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389755(CHEMBL2070093)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389754(CHEMBL2070094)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389765(CHEMBL2070234)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389762(CHEMBL2070099)
Affinity DataIC50:  1.30E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389763(CHEMBL2070232)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389764(CHEMBL2070233)
Affinity DataIC50:  1.60E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389763(CHEMBL2070232)
Affinity DataIC50:  1.60E+3nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389765(CHEMBL2070234)
Affinity DataIC50:  1.70E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389766(CHEMBL2070235)
Affinity DataIC50:  1.80E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389767(CHEMBL2070236)
Affinity DataIC50:  2.10E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389762(CHEMBL2070099)
Affinity DataIC50:  2.40E+3nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389768(CHEMBL2070237)
Affinity DataIC50:  2.40E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389766(CHEMBL2070235)
Affinity DataIC50:  2.50E+3nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389768(CHEMBL2070237)
Affinity DataIC50:  2.50E+3nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389764(CHEMBL2070233)
Affinity DataIC50:  2.60E+3nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389751(CHEMBL2070238)
Affinity DataIC50:  2.80E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389759(CHEMBL2070239)
Affinity DataIC50:  3.20E+3nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389752(CHEMBL2070096)
Affinity DataIC50:  3.30E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389753(CHEMBL2070095)
Affinity DataIC50:  3.40E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389756(CHEMBL2070092)
Affinity DataIC50:  3.50E+3nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM70858(4-mesyl-3-nitro-benzoic acid [2-(1-adamantylamino)...)
Affinity DataIC50:  4.10E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389754(CHEMBL2070094)
Affinity DataIC50:  4.20E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389758(CHEMBL2070090)
Affinity DataIC50:  4.70E+3nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389755(CHEMBL2070093)
Affinity DataIC50:  5.20E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389757(CHEMBL2070091)
Affinity DataIC50:  5.60E+3nMAssay Description:Antagonist activity at human TRalpha assessed as inhibition of interaction with SRC2-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389756(CHEMBL2070092)
Affinity DataIC50:  7.10E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389757(CHEMBL2070091)
Affinity DataIC50:  7.40E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389758(CHEMBL2070090)
Affinity DataIC50:  8.20E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389759(CHEMBL2070239)
Affinity DataIC50:  8.50E+3nMAssay Description:Antagonist activity at human TRbeta assessed as inhibition of interaction with SRC2-2 after 3 hrs by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389759(CHEMBL2070239)
Affinity DataIC50:  3.02E+4nMAssay Description:Antagonist activity at human PPAR-gamma assessed as inhibition of interaction with DRIP-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389753(CHEMBL2070095)
Affinity DataIC50: >6.00E+4nMAssay Description:Antagonist activity at human PPAR-gamma assessed as inhibition of interaction with DRIP-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389751(CHEMBL2070238)
Affinity DataIC50: >6.00E+4nMAssay Description:Antagonist activity at human PPAR-gamma assessed as inhibition of interaction with DRIP-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389760(CHEMBL2070097)
Affinity DataIC50: >6.00E+4nMAssay Description:Antagonist activity at human PPAR-gamma assessed as inhibition of interaction with DRIP-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389761(CHEMBL2070098)
Affinity DataIC50: >6.00E+4nMAssay Description:Antagonist activity at human PPAR-gamma assessed as inhibition of interaction with DRIP-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389762(CHEMBL2070099)
Affinity DataIC50: >6.00E+4nMAssay Description:Antagonist activity at human PPAR-gamma assessed as inhibition of interaction with DRIP-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389763(CHEMBL2070232)
Affinity DataIC50: >6.00E+4nMAssay Description:Antagonist activity at human PPAR-gamma assessed as inhibition of interaction with DRIP-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389764(CHEMBL2070233)
Affinity DataIC50: >6.00E+4nMAssay Description:Antagonist activity at human PPAR-gamma assessed as inhibition of interaction with DRIP-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389765(CHEMBL2070234)
Affinity DataIC50: >6.00E+4nMAssay Description:Antagonist activity at human PPAR-gamma assessed as inhibition of interaction with DRIP-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389766(CHEMBL2070235)
Affinity DataIC50: >6.00E+4nMAssay Description:Antagonist activity at human PPAR-gamma assessed as inhibition of interaction with DRIP-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389767(CHEMBL2070236)
Affinity DataIC50: >6.00E+4nMAssay Description:Antagonist activity at human PPAR-gamma assessed as inhibition of interaction with DRIP-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389768(CHEMBL2070237)
Affinity DataIC50: >6.00E+4nMAssay Description:Antagonist activity at human PPAR-gamma assessed as inhibition of interaction with DRIP-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Institut Pasteur Korea

Curated by ChEMBL
LigandPNGBDBM50389758(CHEMBL2070090)
Affinity DataIC50: >6.00E+4nMAssay Description:Antagonist activity at human PPAR-gamma assessed as inhibition of interaction with DRIP-2 by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 55 total ) | Next | Last >>
Jump to: