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Found 13 Enz. Inhib. hit(s) with all data for entry = 50040043
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50332805((3R,4S,5R,8R,9S,10R,13S,14S)-10,13-Dimethyl-hexade...)
Affinity DataKi:  38nMAssay Description:Inhibition of aromatase in human microsomes using [1beta-3H]androstenedione as substrate after 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50332803((5S,8R,9S,10S,13S,14S)-10,13-dimethyl-5,6,7,8,9,10...)
Affinity DataKi:  50nMAssay Description:Inhibition of aromatase in human microsomes using [1beta-3H]androstenedione as substrate after 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388393(CHEMBL2058266)
Affinity DataKi:  86nMAssay Description:Inhibition of aromatase in human microsomes using [1beta-3H]androstenedione as substrate after 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388396(CHEMBL1077603)
Affinity DataKi:  100nMAssay Description:Inhibition of aromatase in human microsomes using [1beta-3H]androstenedione as substrate after 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388394(CHEMBL2058267)
Affinity DataKi:  9.50E+3nMAssay Description:Inhibition of aromatase in human microsomes using [1beta-3H]androstenedione as substrate after 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50240798((8R,9S,10R,13S,14S)-4-Hydroxy-10,13-dimethyl-1,6,7...)
Affinity DataIC50:  42nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50332807((8R,9S,10R,13S,14S)-10,13-dimethyl-2,3,7,8,9,10,11...)
Affinity DataIC50:  135nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50332805((3R,4S,5R,8R,9S,10R,13S,14S)-10,13-Dimethyl-hexade...)
Affinity DataIC50:  145nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388396(CHEMBL1077603)
Affinity DataIC50:  183nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50332803((5S,8R,9S,10S,13S,14S)-10,13-dimethyl-5,6,7,8,9,10...)
Affinity DataIC50:  225nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388393(CHEMBL2058266)
Affinity DataIC50:  970nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388395(CHEMBL2058268)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388394(CHEMBL2058267)
Affinity DataIC50:  1.73E+3nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed