Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 8340
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
East China University Of Science And Technology

LigandPNGBDBM3175(3-[1-[3-(Amidinothio)propyl]-3-indolyl]-4-(1-methy...)
Affinity DataIC50:  10nMpH: 7.4 T: 2°CAssay Description:The inhibition assays against RSK2 in vitro were determined by ADP Quest® (DiscoveRx) in 96-well flat-bottom plates according to the manufacturer...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
East China University Of Science And Technology

LigandPNGBDBM241956(5-(2-(4-Hydroxyphenyl)hydrazono)pyrimidine-2,4,6(1...)
Affinity DataIC50:  1.95E+3nMpH: 7.4 T: 2°CAssay Description:The inhibition assays against RSK2 in vitro were determined by ADP Quest® (DiscoveRx) in 96-well flat-bottom plates according to the manufacturer...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
East China University Of Science And Technology

LigandPNGBDBM241958(5-(2-(4-Hydroxyphenyl)hydrazono)-dihydro-2-thioxop...)
Affinity DataIC50:  2.19E+3nMpH: 7.4 T: 2°CAssay Description:The inhibition assays against RSK2 in vitro were determined by ADP Quest® (DiscoveRx) in 96-well flat-bottom plates according to the manufacturer...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
East China University Of Science And Technology

LigandPNGBDBM241957(5-(2-(4-Morpholinophenyl)hydrazono)pyrimidine-2,4,...)
Affinity DataIC50:  5.11E+3nMpH: 7.4 T: 2°CAssay Description:The inhibition assays against RSK2 in vitro were determined by ADP Quest® (DiscoveRx) in 96-well flat-bottom plates according to the manufacturer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
East China University Of Science And Technology

LigandPNGBDBM241959(5-(2-(4-Morpholinophenyl)hydrazono-dihydro-2-thiox...)
Affinity DataIC50:  9.23E+3nMpH: 7.4 T: 2°CAssay Description:The inhibition assays against RSK2 in vitro were determined by ADP Quest® (DiscoveRx) in 96-well flat-bottom plates according to the manufacturer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed