Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50039783
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50384053(CHEMBL2032453)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at kappa opioid receptor in guinea pig illeum assessed as electric field-stimulated responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50384054(CHEMBL2032447)
Affinity DataEC50:  3nMAssay Description:Agonist activity at recombinant kappa opioid receptor expressed in human U2OS cells coexpressing beta arrestin/EA complex assessed as beta arrestin r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50384055(CHEMBL2032448)
Affinity DataEC50:  3nMAssay Description:Agonist activity at recombinant kappa opioid receptor expressed in human U2OS cells coexpressing beta arrestin/EA complex assessed as beta arrestin r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50384059(CHEMBL2032452)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at kappa opioid receptor in guinea pig illeum assessed as electric field-stimulated responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50384057(CHEMBL2032450)
Affinity DataEC50:  1.48E+3nMAssay Description:Agonist activity at recombinant kappa opioid receptor expressed in human U2OS cells coexpressing beta arrestin/EA complex assessed as beta arrestin r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50384058(CHEMBL2032451)
Affinity DataEC50:  176nMAssay Description:Agonist activity at recombinant kappa opioid receptor expressed in human U2OS cells coexpressing beta arrestin/EA complex assessed as beta arrestin r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50384054(CHEMBL2032447)
Affinity DataEC50:  0.220nMAssay Description:Agonist activity at kappa opioid receptor in guinea pig illeum assessed as electric field-stimulated responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50384056(CHEMBL2032449)
Affinity DataEC50:  5nMAssay Description:Agonist activity at recombinant kappa opioid receptor expressed in human U2OS cells coexpressing beta arrestin/EA complex assessed as beta arrestin r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed