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Found 22 Enz. Inhib. hit(s) with all data for entry = 50039784
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384076(CHEMBL2029526)
Affinity DataIC50:  5.20E+3nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384074(CHEMBL2029524)
Affinity DataIC50:  1.10E+4nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384073(CHEMBL2029521)
Affinity DataIC50:  1.50E+4nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384060(CHEMBL2029523)
Affinity DataIC50:  3.30E+4nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384075(CHEMBL2029525)
Affinity DataIC50:  3.90E+4nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384062(CHEMBL2029511)
Affinity DataIC50:  5.50E+4nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384064(CHEMBL2029513)
Affinity DataIC50:  6.10E+4nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM51645(6-(4-methoxyphenyl)-1H-thieno[3,2-d]pyrimidin-4-on...)
Affinity DataIC50:  8.60E+4nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM33210(4-(7H-purin-6-yl)morpholine | purine, 9)
Affinity DataIC50:  9.20E+4nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384072(CHEMBL2029520)
Affinity DataIC50:  9.50E+4nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384079(CHEMBL2029522)
Affinity DataIC50:  1.06E+5nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384071(CHEMBL2029519)
Affinity DataIC50:  1.09E+5nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384078(CHEMBL2029517)
Affinity DataIC50:  1.22E+5nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384070(CHEMBL2029518)
Affinity DataIC50:  1.54E+5nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384067(CHEMBL2029516)
Affinity DataIC50:  2.73E+5nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50009126(5-Fluoro-1H-indole-2-carboxylic acid | 5-fluoroind...)
Affinity DataIC50:  2.97E+5nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384065(CHEMBL2029514)
Affinity DataIC50:  3.02E+5nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384066(CHEMBL2029515)
Affinity DataIC50:  4.02E+5nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384069(CHEMBL1877245)
Affinity DataIC50:  4.61E+5nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384063(CHEMBL2029512)
Affinity DataIC50:  4.72E+5nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384077(CHEMBL1891423)
Affinity DataIC50:  4.92E+5nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50384061(CHEMBL2029510)
Affinity DataIC50:  8.28E+5nMAssay Description:Competitive inhibition of PDK1 using [gamma-33P]-ATP as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed