Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50040566
TargetKallikrein-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50396164(CHEMBL2171751)
Affinity DataKi:  8nMAssay Description:Inhibition of human KLK1 using Pro-Phe-Arg-MCA as substrate for 2 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50396166(CHEMBL2171749)
Affinity DataKi:  50nMAssay Description:Inhibition of human KLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50298759((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  65nMAssay Description:Inhibition of human KLK3 using Mu-SRKSQQY-AMC as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50396165(CHEMBL2171750)
Affinity DataKi:  110nMAssay Description:Inhibition of human KLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50396162(CHEMBL2171878)
Affinity DataKi:  300nMAssay Description:Inhibition of KLK3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50396161(CHEMBL2171879)
Affinity DataKi:  500nMAssay Description:Inhibition of KLK3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50396163(CHEMBL2171880)
Affinity DataKi:  1.41E+3nMAssay Description:Inhibition of human KLK2 after 1 hr by phage-display based Immunofluorometric AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed