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Found 34 Enz. Inhib. hit(s) with all data for entry = 50039791
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384195(CHEMBL2029930)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384188(CHEMBL2029923)
Affinity DataKi:  0.580nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384194(CHEMBL2029929)
Affinity DataKi:  0.950nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384190(CHEMBL2029925)
Affinity DataKi:  1.39nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384191(CHEMBL2029926)
Affinity DataKi:  2.26nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384187(CHEMBL2029922)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384189(CHEMBL2029924)
Affinity DataKi:  4.73nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384192(CHEMBL2029927)
Affinity DataKi:  5.78nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384193(CHEMBL2029928)
Affinity DataKi:  7.53nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384186(CHEMBL2029921)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384185(CHEMBL2029920)
Affinity DataKi:  14.2nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384194(CHEMBL2029929)
Affinity DataKi:  29.7nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384196(CHEMBL2029931)
Affinity DataKi:  43.2nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384183(CHEMBL2029918)
Affinity DataKi:  48.6nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384195(CHEMBL2029930)
Affinity DataKi:  48.7nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384182(CHEMBL2029917)
Affinity DataKi:  69.6nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384181(CHEMBL2029916)
Affinity DataKi:  70.7nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384190(CHEMBL2029925)
Affinity DataKi:  82.4nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384181(CHEMBL2029916)
Affinity DataKi:  95.3nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384183(CHEMBL2029918)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384185(CHEMBL2029920)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384182(CHEMBL2029917)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384191(CHEMBL2029926)
Affinity DataKi:  202nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384187(CHEMBL2029922)
Affinity DataKi:  227nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384189(CHEMBL2029924)
Affinity DataKi:  278nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384193(CHEMBL2029928)
Affinity DataKi:  364nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384186(CHEMBL2029921)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384196(CHEMBL2029931)
Affinity DataKi:  478nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384184(CHEMBL2029919)
Affinity DataKi:  483nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384180(CHEMBL2029915)
Affinity DataKi:  903nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384184(CHEMBL2029919)
Affinity DataKi:  2.26E+3nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384192(CHEMBL2029927)
Affinity DataKi:  3.25E+3nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384188(CHEMBL2029923)
Affinity DataKi:  3.58E+3nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50384180(CHEMBL2029915)
Affinity DataKi:  4.19E+3nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed