Affinity DataKi: 7nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 103nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 276nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 661nMAssay Description:Inhibition of M3 muscarinic receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 696nMAssay Description:Inhibition of M2 muscarinic receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 802nMAssay Description:Inhibition of M5 muscarinic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 862nMAssay Description:Inhibition of alpha2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of D2 dopamine receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of M4 muscarinic receptorMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 2.67E+3nMAssay Description:Inhibition of M5 muscarinic receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 2.69E+3nMAssay Description:Inhibition of M5 muscarinic receptorMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 3.83E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 4.24E+3nMAssay Description:Inhibition of alpha2B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.26E+3nMAssay Description:Inhibition of alpha2C adrenergic receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 4.74E+3nMAssay Description:Inhibition of M2 muscarinic receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 5.54E+3nMAssay Description:Inhibition of M1 muscarinic receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 6.17E+3nMAssay Description:Inhibition of M4 muscarinic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.77E+3nMAssay Description:Inhibition of H3 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 7.96E+3nMAssay Description:Inhibition of M1 muscarinic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.91E+3nMAssay Description:Inhibition of D2 dopamine receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of D3 dopamine receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of D5 dopamine receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of D2 dopamine receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of SERTMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of D2 dopamine receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of SERTMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of D2 dopamine receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of D2 dopamine receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of SERTMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of D2 dopamine receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of SERTMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of D2 dopamine receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of alpha1B adrenergic receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of SERTMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of D2 dopamine receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of D2 dopamine receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of D2 dopamine receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of SERTMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL