Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50040110
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50389272(CHEMBL2063565)
Affinity DataIC50:  5.10E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR expressed in Escherichia coli NM522 coexpressing LuxCDABE assessed as inhibition of 3-oxoC6-HSL-induced q...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50389274(CHEMBL2063588)
Affinity DataIC50:  7.40E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR expressed in Escherichia coli NM522 coexpressing LuxCDABE assessed as inhibition of 3-oxoC6-HSL-induced q...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50389277(CHEMBL2063591)
Affinity DataIC50:  8.00E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR expressed in Escherichia coli NM522 coexpressing LuxCDABE assessed as inhibition of 3-oxoC6-HSL-induced q...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50389273(CHEMBL2063594)
Affinity DataIC50:  9.40E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR expressed in Escherichia coli NM522 coexpressing LuxCDABE assessed as inhibition of 3-oxoC6-HSL-induced q...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50389276(CHEMBL2063590)
Affinity DataIC50: >2.00E+5nMAssay Description:Antagonist activity at Vibrio fischeri LuxR expressed in Escherichia coli NM522 coexpressing LuxCDABE assessed as inhibition of 3-oxoC6-HSL-induced q...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50389275(CHEMBL2063589)
Affinity DataIC50: >2.00E+5nMAssay Description:Antagonist activity at Vibrio fischeri LuxR expressed in Escherichia coli NM522 coexpressing LuxCDABE assessed as inhibition of 3-oxoC6-HSL-induced q...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50389278(CHEMBL2063592)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at Vibrio fischeri LuxR expressed in Escherichia coli NM522 coexpressing LuxCDABE assessed as activation of 3-oxoC6-HSL-induced quor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50389279(CHEMBL2063593)
Affinity DataEC50:  3.50E+4nMAssay Description:Agonist activity at Vibrio fischeri LuxR expressed in Escherichia coli NM522 coexpressing LuxCDABE assessed as activation of 3-oxoC6-HSL-induced quor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed