Found 19 Enz. Inhib. hit(s) with all data for entry = 50040666 
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]aldosterone from human mineralocorticoid receptor overexpressed in HEK293 cells by microbeta counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 478nMAssay Description:Displacement of [3H]methyltrienolone from human progesterone receptor overexpressed in HEK293 cells by microbeta counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 669nMAssay Description:Displacement of [3H]dexamethasone from human glucocorticoid receptor overexpressed in HEK293 cells by microbeta counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.17E+3nMAssay Description:Displacement of [3H]-methyltrienolone from human androgen receptor overexpressed in HEK293 cells by microbeta counting assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Antagonist activity at mineralocorticoid receptorMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 7.10nMAssay Description:Displacement of TAMRA-labeled Dexamethasone from human mineralocorticoid receptor expressed in baculovirus infected insect cell lysate after 60 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity against human mineralocorticoid receptor expressed in CHOK1 cells after 10 to 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Competitive antagonist activity at human mineralocorticoid receptor expressed in MR-UAS-bla HEK 293T cells assessed as inhibition of aldosterone-indu...More data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Displacement of [3H]-aldosterone from rat mineralocorticoid receptor after 18 hrs by liquid scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Displacement of [3H]Aldosterone C from rat mineralocorticoid receptor by liquid scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Antagonist activity against human mineralocorticoid receptor expressed in CHOK1 cells after 10 to 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Antagonist activity at mineralocorticoid receptor in human Huh7 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Antagonist activity at mineralocorticoid receptor expressed in african green monkey COS7 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: <500nMAssay Description:Binding affinity to rat mineralocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 510nMAssay Description:Antagonist activity at mineralocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.44E+3nMAssay Description:Antagonist activity against androgen receptor expressed in CHOK1 cells after 10 to 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.47E+3nMAssay Description:Antagonist activity against glucocorticoid receptor expressed in CHOK1 cells after 10 to 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.02E+3nMAssay Description:Antagonist activity against progesterone receptor expressed in CHOK1 cells after 10 to 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at progesterone receptorMore data for this Ligand-Target Pair
