Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 5688
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University Health Science Center

LigandPNGBDBM92622(Benzimidamide, 6d)
Affinity DataIC50:  3.35E+3nMAssay Description:BACE1 inhibitory evaluation was carried out using a Fluorescence Resonance Energy Transfer (FRET) assay kit supplied by PanVera (kit P2985, Madison, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University Health Science Center

LigandPNGBDBM92621(Benzimidamide, 6c)
Affinity DataIC50:  4.36E+3nMAssay Description:BACE1 inhibitory evaluation was carried out using a Fluorescence Resonance Energy Transfer (FRET) assay kit supplied by PanVera (kit P2985, Madison, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University Health Science Center

LigandPNGBDBM92620(Benzimidamide, 6b)
Affinity DataIC50:  7.03E+3nMAssay Description:BACE1 inhibitory evaluation was carried out using a Fluorescence Resonance Energy Transfer (FRET) assay kit supplied by PanVera (kit P2985, Madison, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University Health Science Center

LigandPNGBDBM92619(Benzimidamide, 6a)
Affinity DataIC50:  8.02E+3nMAssay Description:BACE1 inhibitory evaluation was carried out using a Fluorescence Resonance Energy Transfer (FRET) assay kit supplied by PanVera (kit P2985, Madison, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University Health Science Center

LigandPNGBDBM92618(Benzonitrile, 5d)
Affinity DataIC50:  9.35E+3nMAssay Description:BACE1 inhibitory evaluation was carried out using a Fluorescence Resonance Energy Transfer (FRET) assay kit supplied by PanVera (kit P2985, Madison, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University Health Science Center

LigandPNGBDBM92623(Benzonitrile, 8b)
Affinity DataIC50:  9.76E+3nMAssay Description:BACE1 inhibitory evaluation was carried out using a Fluorescence Resonance Energy Transfer (FRET) assay kit supplied by PanVera (kit P2985, Madison, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University Health Science Center

LigandPNGBDBM92617(Benzonitrile, 5c)
Affinity DataIC50:  8.04E+4nMAssay Description:BACE1 inhibitory evaluation was carried out using a Fluorescence Resonance Energy Transfer (FRET) assay kit supplied by PanVera (kit P2985, Madison, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed