Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50040618
TargetVitamin D3 receptor(Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50397074(CHEMBL2171447)
Affinity DataEC50:  1.70nMAssay Description:Transactivation of GAL4-fused VDR ligand binding domain expressed in human HeLa cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  1nMAssay Description:Transactivation of GAL4-fused VDR ligand binding domain expressed in human HeLa cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetVitamin D3 receptor(Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50397073(CHEMBL2171448)
Affinity DataEC50:  5nMAssay Description:Transactivation of GAL4-fused VDR ligand binding domain expressed in human HeLa cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50397077(CHEMBL2171450)
Affinity DataEC50:  0.5nMAssay Description:Transactivation of full length human VDR expressed in human HeLa cells assessed as increase in CYP24 transcription after 18 hrs by luciferase reporte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50397075(CHEMBL2171446)
Affinity DataEC50:  49nMAssay Description:Transactivation of full length human VDR expressed in human HeLa cells assessed as increase in CYP24 transcription after 18 hrs by luciferase reporte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50397074(CHEMBL2171447)
Affinity DataEC50:  2.80nMAssay Description:Transactivation of full length human VDR expressed in human HeLa cells assessed as increase in CYP24 transcription after 18 hrs by luciferase reporte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50397076(CHEMBL2171449)
Affinity DataEC50:  2.20nMAssay Description:Transactivation of full length human VDR expressed in human HeLa cells assessed as increase in CYP24 transcription after 18 hrs by luciferase reporte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  2.5nMAssay Description:Transactivation of full length human VDR expressed in human HeLa cells assessed as increase in CYP24 transcription after 18 hrs by luciferase reporte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank