Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50040242
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391210(CHEMBL2088840)
Affinity DataKi:  17nMAssay Description:Inhibition of CDK9/cyclin-T1 by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391209(CHEMBL2088839)
Affinity DataKi:  28nMAssay Description:Inhibition of CDK1/cyclin B by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391210(CHEMBL2088840)
Affinity DataKi:  53nMAssay Description:Inhibition of CDK1/cyclin B by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391213(CHEMBL2088828)
Affinity DataKi:  55nMAssay Description:Inhibition of CDK1/cyclin B by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391212(CHEMBL2088827)
Affinity DataKi:  61nMAssay Description:Inhibition of CDK1/cyclin B by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391209(CHEMBL2088839)
Affinity DataKi:  91nMAssay Description:Inhibition of CDK9/cyclin-T1 by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391211(CHEMBL2088826)
Affinity DataKi:  96nMAssay Description:Inhibition of CDK1/cyclin B by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391212(CHEMBL2088827)
Affinity DataKi:  98nMAssay Description:Inhibition of CDK9/cyclin-T1 by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391215(CHEMBL2088835)
Affinity DataKi:  127nMAssay Description:Inhibition of CDK1/cyclin B by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391211(CHEMBL2088826)
Affinity DataKi:  140nMAssay Description:Inhibition of CDK9/cyclin-T1 by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391214(CHEMBL2088829)
Affinity DataKi:  154nMAssay Description:Inhibition of CDK9/cyclin-T1 by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391215(CHEMBL2088835)
Affinity DataKi:  176nMAssay Description:Inhibition of CDK9/cyclin-T1 by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391217(CHEMBL2088837)
Affinity DataKi:  207nMAssay Description:Inhibition of CDK9/cyclin-T1 by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391213(CHEMBL2088828)
Affinity DataKi:  253nMAssay Description:Inhibition of CDK9/cyclin-T1 by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391216(CHEMBL2088836)
Affinity DataKi:  285nMAssay Description:Inhibition of CDK9/cyclin-T1 by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391217(CHEMBL2088837)
Affinity DataKi:  287nMAssay Description:Inhibition of CDK1/cyclin B by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391218(CHEMBL2088838)
Affinity DataKi:  314nMAssay Description:Inhibition of CDK9/cyclin-T1 by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391209(CHEMBL2088839)
Affinity DataKi:  328nMAssay Description:Inhibition of CDK7/cyclin-H by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391214(CHEMBL2088829)
Affinity DataKi:  471nMAssay Description:Inhibition of CDK1/cyclin B by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391216(CHEMBL2088836)
Affinity DataKi:  945nMAssay Description:Inhibition of CDK1/cyclin B by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391218(CHEMBL2088838)
Affinity DataKi:  4.53E+3nMAssay Description:Inhibition of CDK1/cyclin B by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391214(CHEMBL2088829)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK7/cyclin-H by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391217(CHEMBL2088837)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK7/cyclin-H by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391212(CHEMBL2088827)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK7/cyclin-H by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391211(CHEMBL2088826)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK7/cyclin-H by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391210(CHEMBL2088840)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK7/cyclin-H by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391215(CHEMBL2088835)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK7/cyclin-H by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391216(CHEMBL2088836)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK7/cyclin-H by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391218(CHEMBL2088838)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK7/cyclin-H by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50391213(CHEMBL2088828)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK7/cyclin-H by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed