Compile Data Set for Download or QSAR
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Found 14 Enz. Inhib. hit(s) with all data for entry = 50040907
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM7781(4-Benzyl-2-methyl-1,2,4-thiadiazolidine-3,5-dione ...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of GSK3beta by kinase-glo assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50401965(PALINURIN)
Affinity DataIC50:  4.50E+3nMAssay Description:Non-ATP competitive inhibition of GSK3betaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50232478(CHEMBL403233)
Affinity DataIC50:  1.02E+4nMAssay Description:Non-ATP competitive inhibition of GSK3betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50401955(CHEMBL2207940)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of GSK3beta by kinase-glo assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50401956(CHEMBL2207939)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of GSK3beta by kinase-glo assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50401966(CHEMBL2207941)
Affinity DataIC50:  4.00E+4nMAssay Description:Non-ATP competitive inhibition of GSK3betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50401960(CHEMBL2207946)
Affinity DataIC50:  4.75E+4nMAssay Description:Inhibition of GSK3beta by kinase-glo assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50401957(CHEMBL2207938)
Affinity DataIC50:  7.72E+4nMAssay Description:Inhibition of GSK3beta by kinase-glo assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50401961(CHEMBL2207945)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GSK3beta by kinase-glo assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50401962(CHEMBL2207944)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GSK3beta by kinase-glo assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50401958(CHEMBL2207947)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GSK3beta by kinase-glo assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50401959(CHEMBL1492321)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GSK3beta by kinase-glo assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50401963(CHEMBL2207943)
Affinity DataIC50:  4.80E+5nMAssay Description:Inhibition of GSK3beta by kinase-glo assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50401964(CHEMBL2207942)
Affinity DataIC50:  8.30E+5nMAssay Description:Inhibition of GSK3beta by kinase-glo assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed