Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Beecham Pharmaceuticals Research Division
Curated by ChEMBL
Beecham Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataKi: 0.590nMAssay Description:Binding affinity for central 5-hydroxytryptamine 3 receptor was determined by displacement of [3H]-ketanserinMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Beecham Pharmaceuticals Research Division
Curated by ChEMBL
Beecham Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for central 5-hydroxytryptamine 3 receptor was determined by displacement of [3H]GR-65630More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Beecham Pharmaceuticals Research Division
Curated by ChEMBL
Beecham Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataKi: <1.00E+4nMAssay Description:5-hydroxytryptamine 3 receptor antagonist activity was confirmed by its ability to antagonize 5-HT evoked tachycardia of rabbit isolated heartMore data for this Ligand-Target Pair