Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50005464
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50492269(CHEMBL594432)
Affinity DataEC50:  32nMAssay Description:Allosteric modulation of human muscarinic M1 acetylcholine receptor expressed CHO cells assessed as intracellular calcium mobilization after 1 hr by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50313638(1-(4-methoxybenzyl)-4-oxo-1,4-dihydroquinoline-3-c...)
Affinity DataEC50:  129nMAssay Description:Allosteric modulation of human muscarinic M1 acetylcholine receptor expressed CHO cells assessed as intracellular calcium mobilization after 1 hr by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50492269(CHEMBL594432)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at human muscarinic M1 acetylcholine receptor expressed CHO cells assessed as intracellular calcium mobilization after 1 hr by Fluo-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed