Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with all data for entry = 50043159
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Henan University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibition of PDK1-mediated Akt activation in human PC3 cells after 2 hrs by Western blotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank