Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50043683
TargetAurora kinase A(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant aurora kinase A (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  1.31E+3nMAssay Description:Inhibition of recombinant ERK1 (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  1.41E+3nMAssay Description:Inhibition of recombinant IKK2 (unknown origin) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50444593(CHEMBL3099835)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant aurora kinase A (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50444595(CHEMBL563560)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant aurora kinase A (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50444593(CHEMBL3099835)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant IKK2 (unknown origin) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50444594(CHEMBL3099832)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant IKK2 (unknown origin) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50444595(CHEMBL563560)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant IKK2 (unknown origin) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50444595(CHEMBL563560)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant ERK1 (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50444594(CHEMBL3099832)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant ERK1 (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50444593(CHEMBL3099835)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant ERK1 (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50444594(CHEMBL3099832)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant aurora kinase A (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed