Compile Data Set for Download or QSAR
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Found 6 Enz. Inhib. hit(s) with all data for entry = 50043447
TargetAromatase(Homo sapiens (Human))
The University Of Tampa

Curated by ChEMBL
LigandPNGBDBM23419((2S)-5,7-dihydroxy-2-(4-hydroxyphenyl)-3,4-dihydro...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of aromatase (unknown origin) using dibenzylfluorescein as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
The University Of Tampa

Curated by ChEMBL
LigandPNGBDBM50441293(3ALPHA,17BETA-DIHYDROXY-5BETA-ANDROSTAN-4-ONE)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of aromatase (unknown origin) using dibenzylfluorescein as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
The University Of Tampa

Curated by ChEMBL
LigandPNGBDBM50441292(CHEMBL2431527)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of aromatase (unknown origin) using dibenzylfluorescein as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
The University Of Tampa

Curated by ChEMBL
LigandPNGBDBM50441295(CHEMBL2431524)
Affinity DataIC50:  2.91E+4nMAssay Description:Inhibition of aromatase (unknown origin) using dibenzylfluorescein as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
The University Of Tampa

Curated by ChEMBL
LigandPNGBDBM50441294(CHEMBL2431525)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibition of aromatase (unknown origin) using dibenzylfluorescein as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
The University Of Tampa

Curated by ChEMBL
LigandPNGBDBM50240798((8R,9S,10R,13S,14S)-4-Hydroxy-10,13-dimethyl-1,6,7...)
Affinity DataIC50:  5.86E+4nMAssay Description:Inhibition of aromatase (unknown origin) using dibenzylfluorescein as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed