Compile Data Set for Download or QSAR
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Found 6 Enz. Inhib. hit(s) with all data for entry = 50044213
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Norwegian Medical Cyclotron Centre

Curated by ChEMBL
LigandPNGBDBM50009298(CHEMBL3233521)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]Triptorelin from rat full-length gonadotropin-releasing hormone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Mus musculus)
Norwegian Medical Cyclotron Centre

Curated by ChEMBL
LigandPNGBDBM50261184(5-((3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaphth...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to mouse gonadotropin-releasing hormone receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Norwegian Medical Cyclotron Centre

Curated by ChEMBL
LigandPNGBDBM50261184(5-((3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaphth...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity to rat gonadotropin-releasing hormone receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Norwegian Medical Cyclotron Centre

Curated by ChEMBL
LigandPNGBDBM50261184(5-((3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaphth...)
Affinity DataKi:  6nMAssay Description:Binding affinity to human gonadotropin-releasing hormone receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Norwegian Medical Cyclotron Centre

Curated by ChEMBL
LigandPNGBDBM50224310(5-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKi:  40nMAssay Description:Binding affinity to human gonadotropin-releasing hormone receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Norwegian Medical Cyclotron Centre

Curated by ChEMBL
LigandPNGBDBM50009297(CHEMBL3233520)
Affinity DataKi:  42nMAssay Description:Displacement of [125I]Triptorelin from rat full-length gonadotropin-releasing hormone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed