Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50044321
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Innsbruck Medical University

Curated by ChEMBL
LigandPNGBDBM50012920(CHEMBL3261356)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of recombinant PKCepsilon (unknown origin)-MBP-tagged RACK2 interaction after 1 hr by ELISA-based assay relative to untreated controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Innsbruck Medical University

Curated by ChEMBL
LigandPNGBDBM50012948(CHEMBL3261358)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of recombinant PKCepsilon (unknown origin)-MBP-tagged RACK2 interaction after 1 hr by ELISA-based assay relative to untreated controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Innsbruck Medical University

Curated by ChEMBL
LigandPNGBDBM50012919(CHEMBL3261343)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of recombinant PKCepsilon (unknown origin)-MBP-tagged RACK2 interaction after 1 hr by ELISA-based assay relative to untreated controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Innsbruck Medical University

Curated by ChEMBL
LigandPNGBDBM50012919(CHEMBL3261343)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of PKCepsilon-induced phosphorylation of Elk1 in human HeLa cells after 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Innsbruck Medical University

Curated by ChEMBL
LigandPNGBDBM50012921(CHEMBL3261337)
Affinity DataIC50:  2.55E+4nMAssay Description:Inhibition of recombinant PKCepsilon (unknown origin)-MBP-tagged RACK2 interaction after 1 hr by ELISA-based assay relative to untreated controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Innsbruck Medical University

Curated by ChEMBL
LigandPNGBDBM50012930(CHEMBL3261357)
Affinity DataIC50:  2.85E+4nMAssay Description:Inhibition of recombinant PKCepsilon (unknown origin)-MBP-tagged RACK2 interaction after 1 hr by ELISA-based assay relative to untreated controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed