Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50044142
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Vit University

Curated by ChEMBL
LigandPNGBDBM50005651(CHEMBL3235427)
Affinity DataIC50:  15nMAssay Description:Inhibition of human DGAT1 using 1,2-diacylglycerol/[14C]-oleoyl CoA as substrate assessed as [14C]-triglyceride formation after 10 mins by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Vit University

Curated by ChEMBL
LigandPNGBDBM50005652(CHEMBL3235428)
Affinity DataIC50:  20nMAssay Description:Inhibition of human DGAT1 using 1,2-diacylglycerol/[14C]-oleoyl CoA as substrate assessed as [14C]-triglyceride formation after 10 mins by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Vit University

Curated by ChEMBL
LigandPNGBDBM50005654(CHEMBL3235430)
Affinity DataIC50:  26nMAssay Description:Inhibition of human DGAT1 using 1,2-diacylglycerol/[14C]-oleoyl CoA as substrate assessed as [14C]-triglyceride formation after 10 mins by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Vit University

Curated by ChEMBL
LigandPNGBDBM50005649(CHEMBL3235425)
Affinity DataIC50:  34nMAssay Description:Inhibition of human DGAT1 using 1,2-diacylglycerol/[14C]-oleoyl CoA as substrate assessed as [14C]-triglyceride formation after 10 mins by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Vit University

Curated by ChEMBL
LigandPNGBDBM50005653(CHEMBL3235429)
Affinity DataIC50:  39nMAssay Description:Inhibition of human DGAT1 using 1,2-diacylglycerol/[14C]-oleoyl CoA as substrate assessed as [14C]-triglyceride formation after 10 mins by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Vit University

Curated by ChEMBL
LigandPNGBDBM50005655(CHEMBL3235431)
Affinity DataIC50:  55nMAssay Description:Inhibition of human DGAT1 using 1,2-diacylglycerol/[14C]-oleoyl CoA as substrate assessed as [14C]-triglyceride formation after 10 mins by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Vit University

Curated by ChEMBL
LigandPNGBDBM50005647(CHEMBL3235422)
Affinity DataIC50:  73nMAssay Description:Inhibition of human DGAT1 using 1,2-diacylglycerol/[14C]-oleoyl CoA as substrate assessed as [14C]-triglyceride formation after 10 mins by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Vit University

Curated by ChEMBL
LigandPNGBDBM50354643(CHEMBL1834206)
Affinity DataIC50:  73nMAssay Description:Inhibition of DGAT1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Vit University

Curated by ChEMBL
LigandPNGBDBM50005648(CHEMBL3235423)
Affinity DataIC50:  76nMAssay Description:Inhibition of human DGAT1 using 1,2-diacylglycerol/[14C]-oleoyl CoA as substrate assessed as [14C]-triglyceride formation after 10 mins by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Vit University

Curated by ChEMBL
LigandPNGBDBM50341782(4-(4-{4-[(2-Phenyl-5-trifluoromethyloxazole-4-carb...)
Affinity DataIC50:  114nMAssay Description:Inhibition of human DGAT1 using 1,2-diacylglycerol/[14C]-oleoyl CoA as substrate assessed as [14C]-triglyceride formation after 10 mins by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Vit University

Curated by ChEMBL
LigandPNGBDBM50005650(CHEMBL3235426)
Affinity DataIC50:  150nMAssay Description:Inhibition of human DGAT1 using 1,2-diacylglycerol/[14C]-oleoyl CoA as substrate assessed as [14C]-triglyceride formation after 10 mins by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed