Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50032825
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335479((R)-N-(1-acetyl-2,2,4-trimethyl-4-(4-(prop-2-ynylo...)
Affinity DataIC50:  39nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335480((R)-N-(1-acetyl-4-(4-((1-(2-(2-(2-azidoethoxy)etho...)
Affinity DataIC50:  324nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335470((R)-4-(3-(2-((1-(2-(2-(2-(4-((4-(1-acetyl-6-biphen...)
Affinity DataIC50:  920nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335472((R)-4-(3-(2-((1-(14-(4-((4-(1-acetyl-6-biphenyl-4-...)
Affinity DataIC50:  1.02E+3nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335471((R)-4-(3-(2-((1-(2-(2-(2-(2-(4-((4-(1-acetyl-6-bip...)
Affinity DataIC50:  1.66E+3nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335473(5-amino-4-(3-(2-((1-(2-(2-(2-azidoethoxy)ethoxy)et...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335474((S)-4-(3-(2-((1-(2-(4-((4-(1-acetyl-6-biphenyl-4-y...)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335475((S)-4-(3-(2-((1-(2-(2-(4-((4-(1-acetyl-6-biphenyl-...)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335476((S)-4-(3-(2-((1-(2-(2-(2-(4-((4-(1-acetyl-6-biphen...)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335477((S)-4-(3-(2-((1-(2-(2-(2-(2-(4-((4-(1-acetyl-6-bip...)
Affinity DataEC50:  57nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335478((S)-4-(3-(2-((1-(14-(4-((4-(1-acetyl-6-biphenyl-4-...)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335467(5-amino-N-tert-butyl-2-(methylthio)-4-(3-(2-oxo-2-...)
Affinity DataEC50:  126nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335473(5-amino-4-(3-(2-((1-(2-(2-(2-azidoethoxy)ethoxy)et...)
Affinity DataEC50:  397nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335472((R)-4-(3-(2-((1-(14-(4-((4-(1-acetyl-6-biphenyl-4-...)
Affinity DataEC50:  55nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335471((R)-4-(3-(2-((1-(2-(2-(2-(2-(4-((4-(1-acetyl-6-bip...)
Affinity DataEC50:  61nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335470((R)-4-(3-(2-((1-(2-(2-(2-(4-((4-(1-acetyl-6-biphen...)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335469((R)-4-(3-(2-((1-(2-(2-(4-((4-(1-acetyl-6-biphenyl-...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335467(5-amino-N-tert-butyl-2-(methylthio)-4-(3-(2-oxo-2-...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335468((R)-4-(3-(2-((1-(2-(4-((4-(1-acetyl-6-biphenyl-4-y...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed