Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50045145
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataKi:  2.10E+4nMAssay Description:Competitive inhibition of Escherichia coli MurD using D-Glu substrate by steady-state enzyme kinetics assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataKi:  2.90E+4nMAssay Description:Partial non-competitive inhibition of Escherichia coli MurD using UMA substrate by steady-state enzyme kinetics assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataKi:  3.90E+4nMAssay Description:Partial un-competitive inhibition of Escherichia coli MurD using ATP substrate by steady-state enzyme kinetics assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramate--L-alanine ligase(Escherichia coli)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of Escherichia coli MurC after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-L-alanyl-D-glutamate--2,6-diaminopimelate ligase(Escherichia coli UMNK88 (Enterobacteria))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046827(CHEMBL3310467)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of Escherichia coli MurE after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramate--L-alanine ligase(Escherichia coli)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046819(CHEMBL3310465)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of Escherichia coli MurC after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of Escherichia coli MurD after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046819(CHEMBL3310465)
Affinity DataIC50:  6.60E+4nMAssay Description:Inhibition of Escherichia coli MurD after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Escherichia coli)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataIC50:  8.90E+4nMAssay Description:Inhibition of Escherichia coli MurF after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-L-alanyl-D-glutamate--2,6-diaminopimelate ligase(Escherichia coli UMNK88 (Enterobacteria))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046819(CHEMBL3310465)
Affinity DataIC50:  8.90E+4nMAssay Description:Inhibition of Escherichia coli MurE after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-L-alanyl-D-glutamate--2,6-diaminopimelate ligase(Escherichia coli UMNK88 (Enterobacteria))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataIC50:  9.30E+4nMAssay Description:Inhibition of Escherichia coli MurE after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046816(CHEMBL3310459)
Affinity DataIC50:  9.50E+4nMAssay Description:Inhibition of Escherichia coli MurD after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Escherichia coli)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046819(CHEMBL3310465)
Affinity DataIC50:  1.02E+5nMAssay Description:Inhibition of Escherichia coli MurF after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramate--L-alanine ligase(Escherichia coli)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046814(CHEMBL3310462)
Affinity DataIC50:  1.07E+5nMAssay Description:Inhibition of Escherichia coli MurC after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramate--L-alanine ligase(Escherichia coli)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046816(CHEMBL3310459)
Affinity DataIC50:  1.33E+5nMAssay Description:Inhibition of Escherichia coli MurC after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046817(CHEMBL3310463)
Affinity DataIC50:  1.68E+5nMAssay Description:Inhibition of Escherichia coli MurD after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046814(CHEMBL3310462)
Affinity DataIC50:  1.70E+5nMAssay Description:Inhibition of Escherichia coli MurD after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramate--L-alanine ligase(Escherichia coli)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046817(CHEMBL3310463)
Affinity DataIC50:  1.72E+5nMAssay Description:Inhibition of Escherichia coli MurC after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Escherichia coli)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046814(CHEMBL3310462)
Affinity DataIC50:  2.01E+5nMAssay Description:Inhibition of Escherichia coli MurF after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramate--L-alanine ligase(Escherichia coli)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046815(CHEMBL3310461)
Affinity DataIC50:  2.05E+5nMAssay Description:Inhibition of Escherichia coli MurC after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046815(CHEMBL3310461)
Affinity DataIC50:  2.06E+5nMAssay Description:Inhibition of Escherichia coli MurD after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-L-alanyl-D-glutamate--2,6-diaminopimelate ligase(Escherichia coli UMNK88 (Enterobacteria))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046824(CHEMBL3310458)
Affinity DataIC50:  2.11E+5nMAssay Description:Inhibition of Escherichia coli MurE after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-L-alanyl-D-glutamate--2,6-diaminopimelate ligase(Escherichia coli UMNK88 (Enterobacteria))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046814(CHEMBL3310462)
Affinity DataIC50:  2.45E+5nMAssay Description:Inhibition of Escherichia coli MurE after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Escherichia coli)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046817(CHEMBL3310463)
Affinity DataIC50:  2.81E+5nMAssay Description:Inhibition of Escherichia coli MurF after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Escherichia coli)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046815(CHEMBL3310461)
Affinity DataIC50:  2.98E+5nMAssay Description:Inhibition of Escherichia coli MurF after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-L-alanyl-D-glutamate--2,6-diaminopimelate ligase(Escherichia coli UMNK88 (Enterobacteria))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046817(CHEMBL3310463)
Affinity DataIC50:  3.03E+5nMAssay Description:Inhibition of Escherichia coli MurE after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-L-alanyl-D-glutamate--2,6-diaminopimelate ligase(Escherichia coli UMNK88 (Enterobacteria))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046823(CHEMBL3310457)
Affinity DataIC50:  3.11E+5nMAssay Description:Inhibition of Escherichia coli MurE after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-L-alanyl-D-glutamate--2,6-diaminopimelate ligase(Escherichia coli UMNK88 (Enterobacteria))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046822(CHEMBL3310456)
Affinity DataIC50:  3.30E+5nMAssay Description:Inhibition of Escherichia coli MurE after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Escherichia coli)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046823(CHEMBL3310457)
Affinity DataIC50:  3.44E+5nMAssay Description:Inhibition of Escherichia coli MurF after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-L-alanyl-D-glutamate--2,6-diaminopimelate ligase(Escherichia coli UMNK88 (Enterobacteria))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046815(CHEMBL3310461)
Affinity DataIC50:  4.94E+5nMAssay Description:Inhibition of Escherichia coli MurE after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed