Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50044664
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM15148(2,3-diphenylquinoxaline 1 | 2-[4-(3-phenylquinoxal...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM15148(2,3-diphenylquinoxaline 1 | 2-[4-(3-phenylquinoxal...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of Akt2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM15148(2,3-diphenylquinoxaline 1 | 2-[4-(3-phenylquinoxal...)
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of Akt3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM15148(2,3-diphenylquinoxaline 1 | 2-[4-(3-phenylquinoxal...)
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of Akt2 PH domain (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM15148(2,3-diphenylquinoxaline 1 | 2-[4-(3-phenylquinoxal...)
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of Akt1 PH domain (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM15148(2,3-diphenylquinoxaline 1 | 2-[4-(3-phenylquinoxal...)
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of SGK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50156074(1,2-bis(3-fluorobenzylidene)hydrazine | CHEMBL3718...)
Affinity DataEC50:  2.60E+3nMAssay Description:Positive allosteric modulator activity at human muscarinic acetylcholine receptor M5 expressed in CHO cells by fluorometric imaging plate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50024542(CHEMBL3334991)
Affinity DataEC50:  33nMAssay Description:Positive allosteric modulator activity at human muscarinic acetylcholine receptor M5 expressed in CHO cells by fluorometric imaging plate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50024560(CHEMBL3334989)
Affinity DataEC50:  3.00E+3nMAssay Description:Negative allosteric modulator activity at human muscarinic acetylcholine receptor M5 expressed in CHO cells by fluorometric imaging plate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50024561(CHEMBL3334990)
Affinity DataEC50:  7.60E+3nMAssay Description:Silent allosteric modulator activity at human muscarinic acetylcholine receptor M5 expressed in CHO cells by fluorometric imaging plate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50024562(CHEMBL2431187)
Affinity DataEC50:  400nMAssay Description:Allosteric agonist activity at human muscarinic acetylcholine receptor M5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed