TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 603nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 813nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 820nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 2.34E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 3.16E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 3.31E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 4.17E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 2.14E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 49nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 32nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 49nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 36nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 263nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 501nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 32nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 324nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 407nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 500nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 260nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 36nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 320nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 96nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 436nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 8nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 410nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 339nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair