Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 6814
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Csir-Central Drug Research Institute

LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)
Affinity DataIC50:  18nMAssay Description:DPP-IV inhibitory activity was determined by measuring the p-nitroaniline (pNA) released from the chromogenic substrate hydrolysis (H-Gly-Pro-pNA). T...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Csir-Central Drug Research Institute

LigandPNGBDBM152800(1-(2-(4-(7-Chloro-4-quinolyl)piperazin-1-yl)acetyl...)
Affinity DataIC50:  3.73E+3nMAssay Description:DPP-IV inhibitory activity was determined by measuring the p-nitroaniline (pNA) released from the chromogenic substrate hydrolysis (H-Gly-Pro-pNA). T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Csir-Central Drug Research Institute

LigandPNGBDBM152801(4-(2-(4-(7-Chloro-4-quinolyl)piperazin-1-yl)acetyl...)
Affinity DataIC50:  5.96E+3nMAssay Description:DPP-IV inhibitory activity was determined by measuring the p-nitroaniline (pNA) released from the chromogenic substrate hydrolysis (H-Gly-Pro-pNA). T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Csir-Central Drug Research Institute

LigandPNGBDBM152799(1-(2-(4-(3-chlorophenyl)piperazin-1-yl)acetyl)pipe...)
Affinity DataIC50:  6.06E+3nMAssay Description:DPP-IV inhibitory activity was determined by measuring the p-nitroaniline (pNA) released from the chromogenic substrate hydrolysis (H-Gly-Pro-pNA). T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Csir-Central Drug Research Institute

LigandPNGBDBM152798(3-(2-(4-(2-Pyridyl)piperazin-1-yl)acetyl)thiazolid...)
Affinity DataIC50:  6.08E+3nMAssay Description:DPP-IV inhibitory activity was determined by measuring the p-nitroaniline (pNA) released from the chromogenic substrate hydrolysis (H-Gly-Pro-pNA). T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed