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Found 34 Enz. Inhib. hit(s) with all data for entry = 50044753
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028620(CHEMBL3342516)
Affinity DataIC50:  33nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028613(CHEMBL3342507)
Affinity DataIC50:  52nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50426581(CHEMBL2324679)
Affinity DataIC50:  58nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028614(CHEMBL3342508)
Affinity DataIC50:  58nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50426580(CHEMBL2324690)
Affinity DataIC50:  68nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028650(CHEMBL3342534)
Affinity DataIC50:  127nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028617(CHEMBL3342511)
Affinity DataIC50:  225nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50021410(CHEMBL3289868)
Affinity DataIC50:  296nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028621(CHEMBL3342517)
Affinity DataIC50:  327nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028616(CHEMBL3342510)
Affinity DataIC50:  380nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028622(CHEMBL3342518)
Affinity DataIC50:  474nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028623(CHEMBL3342522)
Affinity DataIC50:  499nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50021409(CHEMBL3289866)
Affinity DataIC50:  621nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028617(CHEMBL3342511)
Affinity DataIC50:  698nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028615(CHEMBL3342509)
Affinity DataIC50:  715nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028619(CHEMBL3342514)
Affinity DataIC50:  772nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028618(CHEMBL3342513)
Affinity DataIC50:  892nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028626(CHEMBL3342527)
Affinity DataIC50:  1.13E+3nMAssay Description:Displacement of [3H]E2 from human placental microsomal 17beta-HSD2 after 20 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028616(CHEMBL3342510)
Affinity DataIC50:  1.18E+3nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028619(CHEMBL3342514)
Affinity DataIC50:  1.56E+3nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028622(CHEMBL3342518)
Affinity DataIC50:  2.14E+3nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028618(CHEMBL3342513)
Affinity DataIC50:  2.69E+3nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028614(CHEMBL3342508)
Affinity DataIC50:  3.83E+3nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028613(CHEMBL3342507)
Affinity DataIC50:  4.31E+3nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028615(CHEMBL3342509)
Affinity DataIC50:  4.57E+3nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50021409(CHEMBL3289866)
Affinity DataIC50:  4.82E+3nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50426581(CHEMBL2324679)
Affinity DataIC50:  6.73E+3nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50426580(CHEMBL2324690)
Affinity DataIC50:  7.62E+3nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028621(CHEMBL3342517)
Affinity DataIC50:  9.41E+3nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028626(CHEMBL3342527)
Affinity DataIC50:  1.15E+4nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028620(CHEMBL3342516)
Affinity DataIC50:  1.16E+4nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028650(CHEMBL3342534)
Affinity DataIC50:  1.67E+4nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50021410(CHEMBL3289868)
Affinity DataIC50:  1.87E+4nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50028623(CHEMBL3342522)
Affinity DataIC50:  2.53E+4nMAssay Description:Displacement of [3H]E1 from human placental cytosolic17beta-HSD1 after 10 mins by cell-free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed