Compile Data Set for Download or QSAR
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Found 25 Enz. Inhib. hit(s) with all data for entry = 50044831
TargetEstrogen receptor beta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataIC50:  5.60nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERbeta by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataIC50:  5.70nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERalpha by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031809(CHEMBL3360850)
Affinity DataIC50:  8nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERalpha by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031809(CHEMBL3360850)
Affinity DataIC50:  15nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERbeta by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031813(CHEMBL3360847)
Affinity DataIC50:  19nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERbeta by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031813(CHEMBL3360847)
Affinity DataIC50:  40nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERalpha by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM20607((2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethy...)
Affinity DataIC50:  61nMAssay Description:Binding affinity to human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM20607((2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethy...)
Affinity DataIC50:  61nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERalpha by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031811(CHEMBL3360845)
Affinity DataIC50:  140nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERalpha by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031812(CHEMBL3360846)
Affinity DataIC50:  150nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERalpha by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM20607((2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethy...)
Affinity DataIC50:  188nMAssay Description:Binding affinity to human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM20607((2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethy...)
Affinity DataIC50:  190nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERbeta by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031810(CHEMBL3360843)
Affinity DataIC50:  230nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERalpha by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031810(CHEMBL3360843)
Affinity DataIC50:  980nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERbeta by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031812(CHEMBL3360846)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERbeta by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031808(CHEMBL3360844)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERalpha by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031811(CHEMBL3360845)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERbeta by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031808(CHEMBL3360844)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at human recombinant ERalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031814(CHEMBL3360848)
Affinity DataIC50:  1.47E+3nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERalpha by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031808(CHEMBL3360844)
Affinity DataIC50:  4.80E+3nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERbeta by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031816(CHEMBL3360841)
Affinity DataIC50:  1.30E+4nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERalpha by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031815(CHEMBL3360849)
Affinity DataIC50:  1.80E+4nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERalpha by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031814(CHEMBL3360848)
Affinity DataIC50:  2.30E+4nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERbeta by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031816(CHEMBL3360841)
Affinity DataIC50:  5.60E+4nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERbeta by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50031815(CHEMBL3360849)
Affinity DataIC50:  1.44E+5nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERbeta by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed