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Found 6 Enz. Inhib. hit(s) with all data for entry = 6991
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences

LigandPNGBDBM50018011(Aubagio | CHEBI:68540 | HMR-1726 | TERIFLUNOMIDE)
Affinity DataIC50:  64nMpH: 8.0Assay Description:Recombinant human DHODH (final enzyme concentration between 20 and 60 nM in the assay well) were incubated at 37 °C in 50 mM Tris-HCl, 0.1% Triton X-...More data for this Ligand-Target Pair
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences

LigandPNGBDBM163707(Cyclo L-OH-Pro-L-Phe (Fr. 1-4))
Affinity DataIC50:  773nMpH: 8.0Assay Description:Recombinant human DHODH (final enzyme concentration between 20 and 60 nM in the assay well) were incubated at 37 °C in 50 mM Tris-HCl, 0.1% Triton X-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences

LigandPNGBDBM163711(Cyclo L-Pro-L-Val (Fr. 2-1))
Affinity DataIC50: >5.00E+4nMpH: 8.0Assay Description:Recombinant human DHODH (final enzyme concentration between 20 and 60 nM in the assay well) were incubated at 37 °C in 50 mM Tris-HCl, 0.1% Triton X-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences

LigandPNGBDBM163710(Cyclo L-Pro-L-Phe (Fr. 2-2))
Affinity DataIC50: >5.00E+4nMpH: 8.0Assay Description:Recombinant human DHODH (final enzyme concentration between 20 and 60 nM in the assay well) were incubated at 37 °C in 50 mM Tris-HCl, 0.1% Triton X-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences

LigandPNGBDBM163708(Cyclo L-Pro-L-Ile (Fr. 1-5))
Affinity DataIC50: >5.00E+4nMpH: 8.0Assay Description:Recombinant human DHODH (final enzyme concentration between 20 and 60 nM in the assay well) were incubated at 37 °C in 50 mM Tris-HCl, 0.1% Triton X-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences

LigandPNGBDBM163709(Cyclo L-Pro-L-Leu (Fr. 1-6))
Affinity DataIC50: >5.00E+4nMpH: 8.0Assay Description:Recombinant human DHODH (final enzyme concentration between 20 and 60 nM in the assay well) were incubated at 37 °C in 50 mM Tris-HCl, 0.1% Triton X-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed