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Found 7 Enz. Inhib. hit(s) with all data for entry = 6854
TargetC-terminal-binding protein 2(Homo sapiens (Human))
University Of Massachusetts Medical School

LigandPNGBDBM154570(2-Hydroxyimino-3-phenylpropanoic acid (HIPP))
Affinity DataIC50:  745nMpH: 7.1Assay Description:Purified CtBP2 in 50% glycerol was added to 150 μM NADH and variable amounts of MTOB and HIPP in buffer containing 25 mM HEPES, pH 7.1, 25 mM p...More data for this Ligand-Target Pair
TargetC-terminal-binding protein 2(Homo sapiens (Human))
University Of Massachusetts Medical School

LigandPNGBDBM154572(Phenylpyruvate (PPy))
Affinity DataIC50:  1.35E+5nMpH: 7.1Assay Description:Purified CtBP2 in 50% glycerol was added to 150 μM NADH and variable amounts of MTOB and HIPP in buffer containing 25 mM HEPES, pH 7.1, 25 mM p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-terminal-binding protein 1(Homo sapiens (Human))
University Of Massachusetts Medical School

LigandPNGBDBM154570(2-Hydroxyimino-3-phenylpropanoic acid (HIPP))
Affinity DataKd:  2.77E+3nMpH: 8.5Assay Description:Purified CtBP2 was dialyzed overnight against 500 mL of 50 mM glycylglycine at pH 8.5, 300 mM NaCl, 1 mM EDTA, and 2 mM TCEP, with or without 1.5 mM ...More data for this Ligand-Target Pair
TargetC-terminal-binding protein 1(Homo sapiens (Human))
University Of Massachusetts Medical School

LigandPNGBDBM154571(4-Methylthio 2-oxobutyric acid (MTOB))
Affinity DataKd:  1.26E+6nMpH: 7.5Assay Description:Purified CtBP2 was dialyzed overnight against 500 mL of 50 mM glycylglycine at pH 8.5, 300 mM NaCl, 1 mM EDTA, and 2 mM TCEP, with or without 1.5 mM ...More data for this Ligand-Target Pair
TargetC-terminal-binding protein 2(Homo sapiens (Human))
University Of Massachusetts Medical School

LigandPNGBDBM154571(4-Methylthio 2-oxobutyric acid (MTOB))
Affinity DataKd:  2.96E+6nMpH: 8.5Assay Description:Purified CtBP2 was dialyzed overnight against 500 mL of 50 mM glycylglycine at pH 8.5, 300 mM NaCl, 1 mM EDTA, and 2 mM TCEP, with or without 1.5 mM ...More data for this Ligand-Target Pair
TargetC-terminal-binding protein 2(Homo sapiens (Human))
University Of Massachusetts Medical School

LigandPNGBDBM154570(2-Hydroxyimino-3-phenylpropanoic acid (HIPP))
Affinity DataKd:  1.30E+3nMpH: 8.5Assay Description:Purified CtBP2 was dialyzed overnight against 500 mL of 50 mM glycylglycine at pH 8.5, 300 mM NaCl, 1 mM EDTA, and 2 mM TCEP, with or without 1.5 mM ...More data for this Ligand-Target Pair
TargetC-terminal-binding protein 1(Homo sapiens (Human))
University Of Massachusetts Medical School

LigandPNGBDBM154570(2-Hydroxyimino-3-phenylpropanoic acid (HIPP))
Affinity DataKd:  370nMpH: 7.5Assay Description:Purified CtBP2 was dialyzed overnight against 500 mL of 50 mM glycylglycine at pH 8.5, 300 mM NaCl, 1 mM EDTA, and 2 mM TCEP, with or without 1.5 mM ...More data for this Ligand-Target Pair