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Found 5 Enz. Inhib. hit(s) with all data for entry = 50045777
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Rowan University

Curated by ChEMBL
LigandPNGBDBM50351506(CHEMBL1823934)
Affinity DataIC50:  3.00E+4nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Rowan University

Curated by ChEMBL
LigandPNGBDBM50080868(CHEMBL3421670)
Affinity DataEC50:  119nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli BL21 DE3 after 4 to 6 hrs by GFP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Rowan University

Curated by ChEMBL
LigandPNGBDBM50080869(CHEMBL1236450)
Affinity DataEC50:  28nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Rowan University

Curated by ChEMBL
LigandPNGBDBM50080867(CHEMBL3421671)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli BL21 DE3 after 4 to 6 hrs by GFP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Rowan University

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)
Affinity DataEC50:  31nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair