Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50045576
TargetNeurotensin receptor type 2(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50069090(CHEMBL3403506)
Affinity DataKi:  128nMAssay Description:Displacement of [I125]neurotensin from rat NTS2 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50069089(CHEMBL3403505)
Affinity DataKi:  140nMAssay Description:Displacement of [I125]neurotensin from rat NTS2 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50019412(CHEMBL3290096)
Affinity DataKi:  177nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50069091(CHEMBL3403507)
Affinity DataKi:  271nMAssay Description:Displacement of [I125]neurotensin from rat NTS2 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50019417(CHEMBL3290101)
Affinity DataKi:  1.21E+3nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50019423(CHEMBL3290105)
Affinity DataKi:  3.21E+3nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50069092(CHEMBL3403508)
Affinity DataKi:  6.34E+3nMAssay Description:Displacement of [I125]neurotensin from rat NTS2 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50069089(CHEMBL3403505)
Affinity DataKi:  7.18E+3nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50069088(CHEMBL3403504)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50069088(CHEMBL3403504)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [I125]neurotensin from rat NTS2 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50069090(CHEMBL3403506)
Affinity DataKi:  1.02E+4nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50069092(CHEMBL3403508)
Affinity DataKi: >2.50E+4nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50069091(CHEMBL3403507)
Affinity DataKi: >2.50E+4nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50019424(CHEMBL3290106)
Affinity DataKi: >2.50E+4nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50069091(CHEMBL3403507)
Affinity DataEC50:  55nMAssay Description:Agonist activity at rat NTS2 overexpressed in CHO-k1 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50069092(CHEMBL3403508)
Affinity DataEC50:  951nMAssay Description:Agonist activity at rat NTS2 overexpressed in CHO-k1 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed